Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 12805
TargetSerine/threonine-protein kinase ATR(Human)
Jiangsu Yayo Biotechnology Co.

US Patent
LigandPNGBDBM729749(US20250101040, Compound M3)
Affinity DataIC50: 7nMAssay Description:The amount of phosphorylated P53 protein was determined using a time-resolved fluorescence system. Before the starting of the experiment, the followi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Jiangsu Yayo Biotechnology Co.

US Patent
LigandPNGBDBM729750(US20250101040, Compound M7)
Affinity DataIC50: 9nMAssay Description:The amount of phosphorylated P53 protein was determined using a time-resolved fluorescence system. Before the starting of the experiment, the followi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Jiangsu Yayo Biotechnology Co.

US Patent
LigandPNGBDBM729751(US20250101040, Compound M15)
Affinity DataIC50: 10nMAssay Description:The amount of phosphorylated P53 protein was determined using a time-resolved fluorescence system. Before the starting of the experiment, the followi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Jiangsu Yayo Biotechnology Co.

US Patent
LigandPNGBDBM729761(US20250101040, Compound AZD6738)
Affinity DataIC50: 15nMAssay Description:The amount of phosphorylated P53 protein was determined using a time-resolved fluorescence system. Before the starting of the experiment, the followi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Jiangsu Yayo Biotechnology Co.

US Patent
LigandPNGBDBM729758(US20250101040, Compound M19)
Affinity DataIC50: 15nMAssay Description:The amount of phosphorylated P53 protein was determined using a time-resolved fluorescence system. Before the starting of the experiment, the followi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Jiangsu Yayo Biotechnology Co.

US Patent
LigandPNGBDBM729760(US20250101040, Compound M21)
Affinity DataIC50: 22nMAssay Description:The amount of phosphorylated P53 protein was determined using a time-resolved fluorescence system. Before the starting of the experiment, the followi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Jiangsu Yayo Biotechnology Co.

US Patent
LigandPNGBDBM729754(US20250101040, Compound M1a)
Affinity DataIC50: 25nMAssay Description:The amount of phosphorylated P53 protein was determined using a time-resolved fluorescence system. Before the starting of the experiment, the followi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Jiangsu Yayo Biotechnology Co.

US Patent
LigandPNGBDBM729756(US20250101040, Compound M2a)
Affinity DataIC50: 33nMAssay Description:The amount of phosphorylated P53 protein was determined using a time-resolved fluorescence system. Before the starting of the experiment, the followi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Jiangsu Yayo Biotechnology Co.

US Patent
LigandPNGBDBM729759(US20250101040, Compound M20)
Affinity DataIC50: 41nMAssay Description:The amount of phosphorylated P53 protein was determined using a time-resolved fluorescence system. Before the starting of the experiment, the followi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetDNA-dependent protein kinase catalytic subunit(Human)
Jiangsu Yayo Biotechnology Co.

US Patent
LigandPNGBDBM729754(US20250101040, Compound M1a)
Affinity DataIC50: 60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Jiangsu Yayo Biotechnology Co.

US Patent
LigandPNGBDBM729753(US20250101040, Compound M18)
Affinity DataIC50: 64nMAssay Description:The amount of phosphorylated P53 protein was determined using a time-resolved fluorescence system. Before the starting of the experiment, the followi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Jiangsu Yayo Biotechnology Co.

US Patent
LigandPNGBDBM729755(US20250101040, Compound M1b)
Affinity DataIC50: 138nMAssay Description:The amount of phosphorylated P53 protein was determined using a time-resolved fluorescence system. Before the starting of the experiment, the followi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetDNA-dependent protein kinase catalytic subunit(Human)
Jiangsu Yayo Biotechnology Co.

US Patent
LigandPNGBDBM729749(US20250101040, Compound M3)
Affinity DataIC50: 180nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Jiangsu Yayo Biotechnology Co.

US Patent
LigandPNGBDBM729752(US20250101040, Compound M16)
Affinity DataIC50: 445nMAssay Description:The amount of phosphorylated P53 protein was determined using a time-resolved fluorescence system. Before the starting of the experiment, the followi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Jiangsu Yayo Biotechnology Co.

US Patent
LigandPNGBDBM729757(US20250101040, Compound M2b)
Affinity DataIC50: 548nMAssay Description:The amount of phosphorylated P53 protein was determined using a time-resolved fluorescence system. Before the starting of the experiment, the followi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Jiangsu Yayo Biotechnology Co.

US Patent
LigandPNGBDBM729754(US20250101040, Compound M1a)
Affinity DataIC50: 1.00E+4nMAssay Description:Following the experimental methods reported in the reference documents, the test compounds were diluted in a 3-fold series to 0.51 nM (a total of 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Jiangsu Yayo Biotechnology Co.

US Patent
LigandPNGBDBM729749(US20250101040, Compound M3)
Affinity DataIC50: 1.00E+4nMAssay Description:Following the experimental methods reported in the reference documents, the test compounds were diluted in a 3-fold series to 0.51 nM (a total of 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent