Compile Data Set for Download or QSAR
Report error Found 431 Enz. Inhib. hit(s) with all data for entry = 12848
TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733499(US20250115600, Compound 120)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733499(US20250115600, Compound 120)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733498(US20250115600, Compound 119)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733497(US20250115600, Compound 118)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733497(US20250115600, Compound 118)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733502(US20250115600, Compound 123)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

LigandPNGBDBM733501(US20250115600, Compound 122)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733501(US20250115600, Compound 122)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733501(US20250115600, Compound 122)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733500(US20250115600, Compound 121)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733500(US20250115600, Compound 121)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733494(US20250115600, Compound 115)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733493(US20250115600, Compound 114)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733492(US20250115600, Compound 113)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733496(US20250115600, Compound 117)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733495(US20250115600, Compound 116)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733495(US20250115600, Compound 116)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733625(US20250115600, Compound 131)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733588(US20250115600, Compound 130)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733588(US20250115600, Compound 130)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

LigandPNGBDBM733508(US20250115600, Compound 129)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733508(US20250115600, Compound 129)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733508(US20250115600, Compound 129)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733627(US20250115600, Compound 133)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733627(US20250115600, Compound 133)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733626(US20250115600, Compound 132)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733626(US20250115600, Compound 132)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733625(US20250115600, Compound 131)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733502(US20250115600, Compound 123)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733507(US20250115600, Compound 128)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733506(US20250115600, Compound 127)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733506(US20250115600, Compound 127)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733505(US20250115600, Compound 126)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733505(US20250115600, Compound 126)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM50593633(Miransertib | Arq-092 | ARQ 092 | ARQ 092 FREE BAS...)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

LigandPNGBDBM733635(US20250115600, Compound 141)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733635(US20250115600, Compound 141)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733635(US20250115600, Compound 141)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733634(US20250115600, Compound 140)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733634(US20250115600, Compound 140)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733638(US20250115600, Compound B)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733637(US20250115600, Compound A)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-beta serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM50593633(Miransertib | Arq-092 | ARQ 092 | ARQ 092 FREE BAS...)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM50593633(Miransertib | Arq-092 | ARQ 092 | ARQ 092 FREE BAS...)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733630(US20250115600, Compound 136)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733630(US20250115600, Compound 136)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

LigandPNGBDBM733629(US20250115600, Compound 135)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733629(US20250115600, Compound 135)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733629(US20250115600, Compound 135)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Terremoto Biosciences

US Patent
LigandPNGBDBM733633(US20250115600, Compound 139)
Affinity DataIC50: 100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/23/2025
Entry Details
US Patent

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