Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 12969
TargetEpithelial discoidin domain-containing receptor 1(Human)
President and Fellows of Harvard College

US Patent
LigandPNGBDBM744753(US20250177391, Compound 2)
Affinity DataIC50: 9nMAssay Description:DDR1 (h) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKSPGEYVNIEFG (SEQ ID NO: 1), 10 mM magnesium acetate and [γ-33P]-ATP (specific ac...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/30/2025
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
President and Fellows of Harvard College

US Patent
LigandPNGBDBM744728(US20250177391, Compound 1)
Affinity DataIC50: 13nMAssay Description:DDR1 (h) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKSPGEYVNIEFG (SEQ ID NO: 1), 10 mM magnesium acetate and [γ-33P]-ATP (specific ac...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/30/2025
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
President and Fellows of Harvard College

US Patent
LigandPNGBDBM745534(US20250177391, Compound 3)
Affinity DataIC50: 55nMAssay Description:DDR1 (h) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKSPGEYVNIEFG (SEQ ID NO: 1), 10 mM magnesium acetate and [γ-33P]-ATP (specific ac...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/30/2025
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
President and Fellows of Harvard College

US Patent
LigandPNGBDBM746794(US20250177391, Compound 4)
Affinity DataIC50: 66nMAssay Description:DDR1 (h) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKSPGEYVNIEFG (SEQ ID NO: 1), 10 mM magnesium acetate and [γ-33P]-ATP (specific ac...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/30/2025
Entry Details
US Patent

TargetDiscoidin domain-containing receptor 2(Human)
President and Fellows of Harvard College

US Patent
LigandPNGBDBM744753(US20250177391, Compound 2)
Affinity DataIC50: 156nMAssay Description:DDR1 (h) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKSPGEYVNIEFG (SEQ ID NO: 1), 10 mM magnesium acetate and [γ-33P]-ATP (specific ac...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/30/2025
Entry Details
US Patent

TargetDiscoidin domain-containing receptor 2(Human)
President and Fellows of Harvard College

US Patent
LigandPNGBDBM744728(US20250177391, Compound 1)
Affinity DataIC50: 260nMAssay Description:DDR1 (h) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKSPGEYVNIEFG (SEQ ID NO: 1), 10 mM magnesium acetate and [γ-33P]-ATP (specific ac...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/30/2025
Entry Details
US Patent

TargetDiscoidin domain-containing receptor 2(Human)
President and Fellows of Harvard College

US Patent
LigandPNGBDBM746794(US20250177391, Compound 4)
Affinity DataIC50: 1.57E+3nMAssay Description:DDR1 (h) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKSPGEYVNIEFG (SEQ ID NO: 1), 10 mM magnesium acetate and [γ-33P]-ATP (specific ac...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/30/2025
Entry Details
US Patent

TargetDiscoidin domain-containing receptor 2(Human)
President and Fellows of Harvard College

US Patent
LigandPNGBDBM745534(US20250177391, Compound 3)
Affinity DataIC50: 3.30E+3nMAssay Description:DDR1 (h) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKSPGEYVNIEFG (SEQ ID NO: 1), 10 mM magnesium acetate and [γ-33P]-ATP (specific ac...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/30/2025
Entry Details
US Patent