Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 13013
Affinity DataKi: 0.200nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 82nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 82nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 460nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair
Affinity DataKi: 460nMAssay Description:Binding affinities for fentanyl derivatives 1 and 6a-e at KOR, MOR, and DOR were determined by competitive displacement of [3H] diprenorphine as prev...More data for this Ligand-Target Pair



3D Structure (crystal)
