Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 13059
TargetFocal adhesion kinase 1(Human)
Berrybio (Shanghai)

US Patent
LigandPNGBDBM755771(US20250214967, Compound A6)
Affinity DataIC50: 0.390nMAssay Description:The inhibitory activity of a compound against FAK was determined in a buffer containing 5 mM HEPES, pH 7.5, 0.01% Triton, 0.5 mM EGTA, and 0.01% BRIJ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/23/2025
Entry Details
US Patent

TargetFocal adhesion kinase 1(Human)
Berrybio (Shanghai)

US Patent
LigandPNGBDBM755769(N-(1-((1-(2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoiso...)
Affinity DataIC50: 0.400nMAssay Description:The inhibitory activity of a compound against FAK was determined in a buffer containing 5 mM HEPES, pH 7.5, 0.01% Triton, 0.5 mM EGTA, and 0.01% BRIJ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/23/2025
Entry Details
US Patent

TargetFocal adhesion kinase 1(Human)
Berrybio (Shanghai)

US Patent
LigandPNGBDBM755772(US20250214967, Compound A7)
Affinity DataIC50: 0.470nMAssay Description:The inhibitory activity of a compound against FAK was determined in a buffer containing 5 mM HEPES, pH 7.5, 0.01% Triton, 0.5 mM EGTA, and 0.01% BRIJ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/23/2025
Entry Details
US Patent

TargetFocal adhesion kinase 1(Human)
Berrybio (Shanghai)

US Patent
LigandPNGBDBM755770(N-(3-(((2-((4-(4-(4-(2-(2,6-dioxopiperidin-3-yl)-1...)
Affinity DataIC50: 1.80nMAssay Description:The inhibitory activity of a compound against FAK was determined in a buffer containing 5 mM HEPES, pH 7.5, 0.01% Triton, 0.5 mM EGTA, and 0.01% BRIJ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/23/2025
Entry Details
US Patent

TargetFocal adhesion kinase 1(Human)
Berrybio (Shanghai)

US Patent
LigandPNGBDBM755767(N-(3-(((2-(4-(2-(2-(2-((2-(2,6-dioxopiperidin-3-yl...)
Affinity DataIC50: 3nMAssay Description:The inhibitory activity of a compound against FAK was determined in a buffer containing 5 mM HEPES, pH 7.5, 0.01% Triton, 0.5 mM EGTA, and 0.01% BRIJ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/23/2025
Entry Details
US Patent

TargetFocal adhesion kinase 1(Human)
Berrybio (Shanghai)

US Patent
LigandPNGBDBM755766(N-(3-(((2-((4-(2-(2-(2-((2-(2,6-dioxopiperidin-3-y...)
Affinity DataIC50: 4.5nMAssay Description:The inhibitory activity of a compound against FAK was determined in a buffer containing 5 mM HEPES, pH 7.5, 0.01% Triton, 0.5 mM EGTA, and 0.01% BRIJ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/23/2025
Entry Details
US Patent

TargetFocal adhesion kinase 1(Human)
Berrybio (Shanghai)

US Patent
LigandPNGBDBM755768(US20250214967, Compound A3)
Affinity DataIC50: 223nMAssay Description:The inhibitory activity of a compound against FAK was determined in a buffer containing 5 mM HEPES, pH 7.5, 0.01% Triton, 0.5 mM EGTA, and 0.01% BRIJ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/23/2025
Entry Details
US Patent