Compile Data Set for Download or QSAR
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 13145
TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762840((S)—N-(1-cyano-2-(4'-cyano-[1,1'-biphenyl]-4-yl)et...)
Affinity DataIC50: 10nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762860((S)-N-(1-cyano-2-(2-fluoro-4-(1- methyl-2-oxoindol...)
Affinity DataIC50: 10nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762859((S)-N-(1-cyano-2-(2-fluoro-4- (1'-(oxetan-3-yl)-3H...)
Affinity DataIC50: 10nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762861((S)-N-(1-cyano-2-(2-fluoro-4-(1- methyl-2-oxoindol...)
Affinity DataIC50: 10nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762832((S)-N-(1-cyano-2-(2-fluoro-4-(1- methyl-2-oxoindol...)
Affinity DataIC50: 10nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762848((S)—N-(1-cyano-2-(2-fluoro-4-(3-methyl-2-oxo-2,3-d...)
Affinity DataIC50: 10nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762831((S)—N-(1-cyano-2-(2-fluoro-4-(1'-(oxetan-3-yl)-3H-...)
Affinity DataIC50: 10nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762847((S)-N-(1-cyano-2-(2-fluoro-4-(3- methyl-2-oxo-2,3-...)
Affinity DataIC50: 10nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762863((S)-N-(1-cyano-2-(2-fluoro-4-(1- methyl-2-oxoindol...)
Affinity DataIC50: 10nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762853((S)-N-(1-cyano-2-(4'-cyano-3- fluoro-[1,1'-bipheny...)
Affinity DataIC50: 10nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762856(Single enantiomers of N-(1-cyano-2-(5-(4-cyanophen...)
Affinity DataIC50: 55nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762855(N-(1-cyano-2-(5-(4- cyanophenyl)-3-fluoropyridin-2...)
Affinity DataIC50: 55nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762828((S)-N-(1-cyano-2-(4'-cyano-3- fluoro-[1,1'-bipheny...)
Affinity DataIC50: 55nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762827((S)-N-(1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4-yl)e...)
Affinity DataIC50: 55nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762830((S)—N-(1-cyano-2-(4-(3-methyl-2-oxo-2,3-dihydroben...)
Affinity DataIC50: 55nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762829((S)-N-(1-cyano-2-(4'-cyano-3- fluoro-[1,1'-bipheny...)
Affinity DataIC50: 55nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762850((S)-N-(1-cyano-2-(2-fluoro-4- (1'-(oxetan-3-yl)-3H...)
Affinity DataIC50: 55nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762849((S)-N-(1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4-yl)e...)
Affinity DataIC50: 55nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762852((S)-N-(1-cyano-2-(4'-cyano-3- fluoro-[1,1'-bipheny...)
Affinity DataIC50: 55nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762834((S)-N-(1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4-yl)e...)
Affinity DataIC50: 55nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762866((S)-N-(1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4-yl)e...)
Affinity DataIC50: 55nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762833((S)—N-(1-cyano-2-(4'-cyano-[1,1'-biphenyl]-4-yl)et...)
Affinity DataIC50: 55nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762868((S)-N-(1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4-yl)e...)
Affinity DataIC50: 55nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762867((S)-N-(1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4-yl)e...)
Affinity DataIC50: 55nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762838((S)-N-(1-cyano-2-(4-(1-methyl- 2-oxoindolin-6-yl)p...)
Affinity DataIC50: 55nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762842((S)-N-(1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4-yl)e...)
Affinity DataIC50: 550nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762825((S)—N-(1-cyano-2-(4'-cyano-[1,1'-biphenyl]-4-yl)et...)
Affinity DataIC50: 550nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762846((S)-N-(1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4-yl)e...)
Affinity DataIC50: 550nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762862((S)-N-(1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4-yl)e...)
Affinity DataIC50: 550nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762845(N-((S)-1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4-yl)e...)
Affinity DataIC50: 550nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762865((S)-N-(1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4-yl)e...)
Affinity DataIC50: 550nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762835((S)-N-(1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4-yl)e...)
Affinity DataIC50: 550nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762854(N-(1-cyano-2-(5-(4-cyanophenyl)-3-fluoropyridin-2-...)
Affinity DataIC50: 550nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762869((S)-N-(1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4- yl)...)
Affinity DataIC50: 550nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762839((S)—N-(1-cyano-2-(4'-cyano-[1,1'-biphenyl]-4-yl)et...)
Affinity DataIC50: 5.50E+3nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762826((S)-N-(1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4-yl)e...)
Affinity DataIC50: 5.50E+3nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762858((S)—N-(1-cyano-2-(4'-cyano-[1,1'-biphenyl]-4-yl)et...)
Affinity DataIC50: 5.50E+3nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762841((S)-N-(1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4-yl)e...)
Affinity DataIC50: 5.50E+3nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762857(Enantiomer 2 of N-(1-cyano-2- (5-(4-cyanophenyl)-3...)
Affinity DataIC50: 5.50E+3nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762844((S)-N-(1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4-yl)e...)
Affinity DataIC50: 5.50E+3nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762843(N-((S)-1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4-yl)e...)
Affinity DataIC50: 5.50E+3nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762864((S)-N-(1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4-yl)e...)
Affinity DataIC50: 5.50E+3nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762836((S)-3-Benzyl-N-(1-cyano-2-(4'-cyano-[1,1'-biphenyl...)
Affinity DataIC50: 5.50E+3nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762851(N-((S)-1-cyano-2-(4'-cyano- [1,1'-biphenyl]-4-yl)e...)
Affinity DataIC50: 5.50E+3nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762837((S)—N-(1-cyano-2-(4'-cyano-[1,1'-biphenyl]-4-yl)et...)
Affinity DataIC50: 5.50E+3nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent