Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 13168
LigandPNGBDBM764595(US20250257055, Example 33 | US20250263415, Example...)
Affinity DataIC50: 0.200nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764596(US20250257055, Example 34 | US20250263415, Example...)
Affinity DataIC50: 0.200nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764573(US20250257055, Example 10 | US20250263415, Example...)
Affinity DataIC50: 0.400nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764594(US20250257055, Example 32 | US20250263415, Example...)
Affinity DataIC50: 0.400nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764567(US20250257055, Example 4 | US20250263415, Example ...)
Affinity DataIC50: 0.5nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764572(US20250257055, Example 9 | US20250263415, Example ...)
Affinity DataIC50: 0.600nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764566(US20250257055, Example 3 | US20250263415, Example ...)
Affinity DataIC50: 0.600nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764570(US20250257055, Example 7 | US20250263415, Example ...)
Affinity DataIC50: 0.900nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764593(US20250257055, Example 31 | US20250263415, Example...)
Affinity DataIC50: 1nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764574(US20250257055, Example 11 | US20250263415, Example...)
Affinity DataIC50: 2nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764592(US20250257055, Example 30 | US20250263415, Example...)
Affinity DataIC50: 2nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764580(US20250257055, Example 17 | US20250263415, Example...)
Affinity DataIC50: 2nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM764583(US20250257055, Example 20 | US20250263415, Example...)
Affinity DataIC50: 2nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764591(US20250257055, Example 29 | US20250263415, Example...)
Affinity DataIC50: 3nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764576(US20250257055, Example 13 | US20250263415, Example...)
Affinity DataIC50: 5nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764597(US20250257055, Example 35 | US20250263415, Example...)
Affinity DataIC50: 5nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764588(US20250257055, Example 25 | US20250263415, Example...)
Affinity DataIC50: 6nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764575(US20250257055, Example 12 | US20250263415, Example...)
Affinity DataIC50: 6nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764578(US20250257055, Example 15 | US20250263415, Example...)
Affinity DataIC50: 6nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764568(US20250257055, Example 5 | US20250263415, Example ...)
Affinity DataIC50: 6nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764590(US20250257055, Example 27 | US20250263415, Example...)
Affinity DataIC50: 7nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764582(US20250257055, Example 19)
Affinity DataIC50: 7nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764589(US20250257055, Example 26 | US20250263415, Example...)
Affinity DataIC50: 9nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764586(US20250257055, Example 23 | US20250263415, Example...)
Affinity DataIC50: 9nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764587(US20250257055, Example 24 | US20250263415, Example...)
Affinity DataIC50: 10nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764585(US20250257055, Example 22 | US20250263415, Example...)
Affinity DataIC50: 11nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764564(N-[(4-fluorophenyl)methyl]-2-[(1'S)-5'-{1-[1-(oxet...)
Affinity DataIC50: 16nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764571(US20250257055, Example 8 | US20250263415, Example ...)
Affinity DataIC50: 17nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764565(US20250257055, Example 2)
Affinity DataIC50: 19nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764569(US20250257055, Example 6 | US20250263415, Example ...)
Affinity DataIC50: 20nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764584(US20250257055, Example 21 | US20250263415, Example...)
Affinity DataIC50: 52nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764579(US20250257055, Example 16 | US20250263415, Example...)
Affinity DataIC50: 54nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764581(US20250257055, Example 18 | US20250263415, Example...)
Affinity DataIC50: 58nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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LigandPNGBDBM764577(US20250257055, Example 14 | US20250263415, Example...)
Affinity DataIC50: 124nMAssay Description:The HAT activity inhibitory ability of HAT inhibitors was evaluated using SensoLyte HAT(p300) Assay Kit (ANASPEC, AS-72172). Specifically, 7.5 μL of ...More data for this Ligand-Target Pair
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