Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 13192
TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765942(2,5-dichloro-N- (3-(2-(((1R,4R)-4- (dimethylamino)...)
Affinity DataIC50: 1.11nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765946(N-(3-(2- (((1R,4R)-4- aminocyclohexyl) amino)quina...)
Affinity DataIC50: 1.64nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765924((1R,3R)-3-((6-(3- ((2,5-dichloro-3- (hydroxymethyl...)
Affinity DataIC50: 2.12nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765945(5-chloro-N-(3-(2- (((1R,4R)-4- (dimethylamino)cy- ...)
Affinity DataIC50: 2.35nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765918(2,5-dichloro-N- (2,4-difluoro-3- (2-(((1R,3R)-3- (...)
Affinity DataIC50: 2.63nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765940(5-chloro-N-(2,4- difluoro-3-(2- (((1R,4R)-4- (meth...)
Affinity DataIC50: 3.23nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765922(5-chloro-N-(3-(2- (((1R,4R)-4- (dimethylamino)cy- ...)
Affinity DataIC50: 3.36nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765927((1R,3R)-3-((6-(3- ((5-chloro-2- methoxypyridine)- ...)
Affinity DataIC50: 3.39nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765920((1R,4R)-4-((6-(3- ((2,5-dichloro-3- (hydroxymethyl...)
Affinity DataIC50: 3.94nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765944(5-chloro-N-(3-(2- (((1R,4R)-4- (dimethylamino)cy- ...)
Affinity DataIC50: 3.95nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765926(5-chloro-N-(2,4- difluoro-3-(2- (((1R,3R)-3-(((2- ...)
Affinity DataIC50: 3.96nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765928((2R,4S)-4-((6-(3- ((5-chloro-2- methoxypyridine)- ...)
Affinity DataIC50: 4.18nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765941(N-(3-(2- (((1R,4R)-4- aminocyclohexyl) amino)-8- e...)
Affinity DataIC50: 5.13nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765919((2R,4S)-4-((6-(3- ((2,5-dichloro-3- (hydroxymethyl...)
Affinity DataIC50: 5.43nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765934(5-chloro-N-(3-(2- ((1,1- dioxidotetrahydro- thioph...)
Affinity DataIC50: 6.66nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765937(N-(4-(2-amino-8- ethylquinazolin- 6-yl)-3,5- diflu...)
Affinity DataIC50: 7.32nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765925(2,5-dichloro-N- (3-(2-((1,1- dioxidotetrahydro- th...)
Affinity DataIC50: 7.62nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765938(N-(4-(2-amino-8- ethylquinazolin- 6-yl)-3,5- dichl...)
Affinity DataIC50: 8.33nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765936(N-(4-(2-amino-8- ethylquinazolin- 6-yl)-3,5- dichl...)
Affinity DataIC50: 8.82nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765930((2R,4S)-4-((6- (2,6-dichloro-3- ((5-chloro-2- meth...)
Affinity DataIC50: 9.17nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765932((1R,4R)-4-((6-(3- ((5-chloro-2- methoxypyridine)- ...)
Affinity DataIC50: 10.2nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765917((R)-3-((6-(3- ((2,5-dichloro-3- (hydroxymethyl)phe...)
Affinity DataIC50: 10.4nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765921((R)-3-((6-(3-((5- chloro-2- methoxypyridine)- 3-su...)
Affinity DataIC50: 11.4nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765929((1R,3R)-3-((6- (2,6-dichloro-3- ((5-chloro-2- meth...)
Affinity DataIC50: 11.7nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765923(5-chloro-N-(2,4- dichloro-3-(2- (((1R,3R)-3-(((2- ...)
Affinity DataIC50: 12.6nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765953(N-(4-(2- aminoquinazolin- 6-yl)-3,5- dichloropyrid...)
Affinity DataIC50: 19.4nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765935(5-chloro-N-(2,4- dichloro-3-(2- ((1,1- dioxidotetr...)
Affinity DataIC50: 25.3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765947(2-chloro-N-(3-(2- (((1R,4R)-4- (dimethylamino)cy- ...)
Affinity DataIC50: 26.8nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765933((1R,4R)-4-((6- (2,6-dichloro-3- ((5-chloro-2- meth...)
Affinity DataIC50: 31.9nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765943((1R,3R)-3-((6-(3- ((5-chloro-2- methoxypyridine)- ...)
Affinity DataIC50: 34.3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765950(N-(3-(2- (((1R,4R)-4- aminocyclohexyl) amino)-8- e...)
Affinity DataIC50: 39.8nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765931((R)-3-((6-(2,6- dichloro-3-((5- chloro-2- methoxyp...)
Affinity DataIC50: 41.6nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765948(2-chloro-N-(3-(8- ethyl-2-(((1R,4R)- 4- (methylami...)
Affinity DataIC50: 43.7nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765949(2-chloro-N-(2,4- difluoro-3-(2- (((1R,4R)-4- (meth...)
Affinity DataIC50: 63.2nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765951(2-chloro-N-(3-(2- (((1R,4R)-4- (dimethylamino)cy- ...)
Affinity DataIC50: 81.2nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765939(5-chloro-N-(3-(8- ethyl-2-(((1R,4R)- 4- (methylami...)
Affinity DataIC50: 88.3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765952(N-(3-(2- (((1R,4R)-4- aminocyclohexyl) amino)quina...)
Affinity DataIC50: 123nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)TBA
LigandPNGBDBM765954(N-(4-(2- aminoquinazolin- 6-yl)-3,5- difluoropyrid...)
Affinity DataIC50: 367nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent