Compile Data Set for Download or QSAR
Report error Found 47 Enz. Inhib. hit(s) with all data for entry = 13213
LigandPNGBDBM767370(5-[6-[2-(3-pyridylmethyl)quinuclidin-3-yl]oxypyrid...)
Affinity DataKi:  1nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767379(US20250270203, Compound 2S,3R-11)
Affinity DataKi:  1nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767378(2-(1H-indol-5-yl)-5-[2-(3-pyridylmethyl) quinuclid...)
Affinity DataKi:  1.40nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767372(2-(1H-indol-5-yl)-5-[2-(3-pyridylmethyl)quinuclidi...)
Affinity DataKi:  11nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767385(2-(3-pyridylmethyl)-3-[6-(1H-pyrrol-2-yl)pyridazin...)
Affinity DataKi:  11.1nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767376(5-[6-[2-(3-pyridylmethyl) quinuclidin-3-yl]oxy-3-p...)
Affinity DataKi:  17.3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767383(6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1,...)
Affinity DataKi:  18.8nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767373(6-[6-[2-(3-pyridylmethyl)quinuclidin-3-yl]oxypyrid...)
Affinity DataKi:  19nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767381(US20250270203, Compound 2R,3S-11)
Affinity DataKi:  34nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767374(2-(3-pyridylmethyl)-3-[6-(1H-pyrrol-2-yl)pyridazin...)
Affinity DataKi:  42nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767384(6-[6-[2-(3-pyridylmethyl) quinuclidin-3-yl]oxypyri...)
Affinity DataKi:  42nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767383(6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1,...)
Affinity DataKi:  50nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767375(2-(3-pyridylmethyl) quinuclidin-3-ol | US202502702...)
Affinity DataKi:  58nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767369(5-[6-[2-(3-pyridylmethyl)quinuclidin-3-yl]oxy-3-py...)
Affinity DataKi:  58nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767376(5-[6-[2-(3-pyridylmethyl) quinuclidin-3-yl]oxy-3-p...)
Affinity DataKi:  59nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767378(2-(1H-indol-5-yl)-5-[2-(3-pyridylmethyl) quinuclid...)
Affinity DataKi:  73nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767379(US20250270203, Compound 2S,3R-11)
Affinity DataKi:  77nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767388(3-[2-(3-pyridylmethyl) quinuclidin-3-yl]oxyisoquin...)
Affinity DataKi:  100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767367(3-(6-phenylpyridazin-3-yl)oxy-2-(3-pyridylmethyl)q...)
Affinity DataKi:  100nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767388(3-[2-(3-pyridylmethyl) quinuclidin-3-yl]oxyisoquin...)
Affinity DataKi:  120nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767387(2-[2-(3-pyridylmethyl) quinuclidin-3-yl]oxyquinoli...)
Affinity DataKi:  140nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767376(5-[6-[2-(3-pyridylmethyl) quinuclidin-3-yl]oxy-3-p...)
Affinity DataKi:  200nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767384(6-[6-[2-(3-pyridylmethyl) quinuclidin-3-yl]oxypyri...)
Affinity DataKi:  200nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767385(2-(3-pyridylmethyl)-3-[6-(1H-pyrrol-2-yl)pyridazin...)
Affinity DataKi:  220nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767377(5-[5-[2-(3-pyridylmethyl) quinuclidin-3-yl]oxypyra...)
Affinity DataKi:  230nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767377(5-[5-[2-(3-pyridylmethyl) quinuclidin-3-yl]oxypyra...)
Affinity DataKi:  240nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767371(5-[5-[2-(3-pyridylmethyl)quinuclidin-3-yl]oxypyraz...)
Affinity DataKi:  240nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767368(2-phenyl-5-[2-(3-pyridylmethyl)quinuclidin-3-yl]ox...)
Affinity DataKi:  320nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767389(3-(6-imidazol-1-ylpyridazin-3-yl)oxy-2-(3-pyridylm...)
Affinity DataKi:  320nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767389(3-(6-imidazol-1-ylpyridazin-3-yl)oxy-2-(3-pyridylm...)
Affinity DataKi:  330nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767389(3-(6-imidazol-1-ylpyridazin-3-yl)oxy-2-(3-pyridylm...)
Affinity DataKi:  340nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767377(5-[5-[2-(3-pyridylmethyl) quinuclidin-3-yl]oxypyra...)
Affinity DataKi:  400nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767385(2-(3-pyridylmethyl)-3-[6-(1H-pyrrol-2-yl)pyridazin...)
Affinity DataKi:  440nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767375(2-(3-pyridylmethyl) quinuclidin-3-ol | US202502702...)
Affinity DataKi:  470nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767381(US20250270203, Compound 2R,3S-11)
Affinity DataKi:  730nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767378(2-(1H-indol-5-yl)-5-[2-(3-pyridylmethyl) quinuclid...)
Affinity DataKi:  730nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767384(6-[6-[2-(3-pyridylmethyl) quinuclidin-3-yl]oxypyri...)
Affinity DataKi:  730nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767375(2-(3-pyridylmethyl) quinuclidin-3-ol | US202502702...)
Affinity DataKi:  780nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767379(US20250270203, Compound 2S,3R-11)
Affinity DataKi:  780nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767387(2-[2-(3-pyridylmethyl) quinuclidin-3-yl]oxyquinoli...)
Affinity DataKi:  800nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767388(3-[2-(3-pyridylmethyl) quinuclidin-3-yl]oxyisoquin...)
Affinity DataKi:  800nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767386(6-fluoro-2-[2-(3-pyridylmethyl) quinuclidin-3-yl]o...)
Affinity DataKi:  1.00E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767383(6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1,...)
Affinity DataKi:  1.08E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767381(US20250270203, Compound 2R,3S-11)
Affinity DataKi:  1.21E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767386(6-fluoro-2-[2-(3-pyridylmethyl) quinuclidin-3-yl]o...)
Affinity DataKi:  1.87E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767386(6-fluoro-2-[2-(3-pyridylmethyl) quinuclidin-3-yl]o...)
Affinity DataKi:  2.15E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM767387(2-[2-(3-pyridylmethyl) quinuclidin-3-yl]oxyquinoli...)
Affinity DataKi:  2.92E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent