Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 13373
TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784327(US20250340530, Example 8)
Affinity DataKi:  1.40nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784338(US20250340530, Example 19)
Affinity DataKi:  1.5nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784326(US20250340530, Example 7)
Affinity DataKi:  1.60nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784331(US20250340530, Example 12)
Affinity DataKi:  1.60nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784320(US20250340530, Example 1)
Affinity DataKi:  1.70nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784329(US20250340530, Example 10)
Affinity DataKi:  1.90nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784324(US20250340530, Example 5)
Affinity DataKi:  1.90nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784351(US20250340530, Comparative Example 1)
Affinity DataKi:  1.90nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784330(US20250340530, Example 11)
Affinity DataKi:  1.90nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784333(US20250340530, Example 14)
Affinity DataKi:  2nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784323(US20250340530, Example 4)
Affinity DataKi:  2.20nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784321(US20250340530, Example 2)
Affinity DataKi:  2.20nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784342(US20250340530, Example 23)
Affinity DataKi:  2.30nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784325(US20250340530, Example 6)
Affinity DataKi:  2.40nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784350(US20250340530, Example 31)
Affinity DataKi:  2.5nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784344(US20250340530, Example 25)
Affinity DataKi:  2.60nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784337(US20250340530, Example 18)
Affinity DataKi:  2.60nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784332(US20250340530, Example 13)
Affinity DataKi:  2.60nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784336(US20250340530, Example 17)
Affinity DataKi:  3nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784341(US20250340530, Example 22)
Affinity DataKi:  3.30nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784334(US20250340530, Example 15)
Affinity DataKi:  3.40nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784335(US20250340530, Example 16)
Affinity DataKi:  3.40nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784339(US20250340530, Example 20)
Affinity DataKi:  3.70nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784340(US20250340530, Example 21)
Affinity DataKi:  3.90nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784343(US20250340530, Example 24)
Affinity DataKi:  4.40nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784328(US20250340530, Example 9)
Affinity DataKi:  4.5nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784346(US20250340530, Example 27)
Affinity DataKi:  4.70nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784322(US20250340530, Example 3)
Affinity DataKi:  4.90nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784352(US20250340530, Comparactive Example 3)
Affinity DataKi:  4.90nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784345(US20250340530, Example 26)
Affinity DataKi:  7nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784349(US20250340530, Example 30)
Affinity DataKi:  8.60nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784347(US20250340530, Example 28)
Affinity DataKi:  17.7nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM784348(US20250340530, Example 29)
Affinity DataKi:  19nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/25/2026
Entry Details US Patent