Compile Data Set for Download or QSAR
Report error Found 84 Enz. Inhib. hit(s) with all data for entry = 13380
TargetProto-oncogene tyrosine-protein kinase Src(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM31089(DASATINIB | US20250340886, Compound A8)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent
PDB3D3D Structure (crystal)
TargetTyrosine-protein kinase ABL1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM31089(DASATINIB | US20250340886, Compound A8)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK3(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM31089(DASATINIB | US20250340886, Compound A8)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK2(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM31089(DASATINIB | US20250340886, Compound A8)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM31089(DASATINIB | US20250340886, Compound A8)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK3(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784726(N-(2,6-dichlorophenyl)-2- ((6-(4-(2- hydroxyethyl)...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK2(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784726(N-(2,6-dichlorophenyl)-2- ((6-(4-(2- hydroxyethyl)...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784726(N-(2,6-dichlorophenyl)-2- ((6-(4-(2- hydroxyethyl)...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK3(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784728(N-(2,6-dibromophenyl)-2- ((6-(4-(2-hydroxyethyl)pi...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK2(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784728(N-(2,6-dibromophenyl)-2- ((6-(4-(2-hydroxyethyl)pi...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784728(N-(2,6-dibromophenyl)-2- ((6-(4-(2-hydroxyethyl)pi...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784727(N-(2-bromo-6-chlorophenyl)-2- ((6-(4-(2-hydroxyeth...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetTyrosine-protein kinase ABL1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784727(N-(2-bromo-6-chlorophenyl)-2- ((6-(4-(2-hydroxyeth...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK3(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784727(N-(2-bromo-6-chlorophenyl)-2- ((6-(4-(2-hydroxyeth...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK2(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784727(N-(2-bromo-6-chlorophenyl)-2- ((6-(4-(2-hydroxyeth...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784727(N-(2-bromo-6-chlorophenyl)-2- ((6-(4-(2-hydroxyeth...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM50506980(CHEMBL4583196 | US20250340886, Compound A10)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK3(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784721(2-((6-(4-(2-hydroxyethyl)piperazin- 1-yl)-2- methy...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK2(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784721(2-((6-(4-(2-hydroxyethyl)piperazin- 1-yl)-2- methy...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784721(2-((6-(4-(2-hydroxyethyl)piperazin- 1-yl)-2- methy...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK3(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM31089(DASATINIB | US20250340886, Compound A8)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK2(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM31089(DASATINIB | US20250340886, Compound A8)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM31089(DASATINIB | US20250340886, Compound A8)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK3(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784725(N-(2,6-dimethylphenyl)-2- ((6-(4-(2- hydroxyethyl)...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK2(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784725(N-(2,6-dimethylphenyl)-2- ((6-(4-(2- hydroxyethyl)...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784725(N-(2,6-dimethylphenyl)-2- ((6-(4-(2- hydroxyethyl)...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK2(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784723(((6-(4-(2-hydroxyethyl)piperazin- 1-yl)-2- methylp...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784723(((6-(4-(2-hydroxyethyl)piperazin- 1-yl)-2- methylp...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK3(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM50506980(CHEMBL4583196 | US20250340886, Compound A10)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK2(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM50506980(CHEMBL4583196 | US20250340886, Compound A10)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK2(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM13277(N-(2-Chloro-6-methylphenyl)-2-(6-(2-hydroxyethylam...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM13277(N-(2-Chloro-6-methylphenyl)-2-(6-(2-hydroxyethylam...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784732(2-((6-(4-acetylpiperazin-1-yl)- 2-methylpyrimidin-...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetTyrosine-protein kinase ABL1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784732(2-((6-(4-acetylpiperazin-1-yl)- 2-methylpyrimidin-...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK3(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784732(2-((6-(4-acetylpiperazin-1-yl)- 2-methylpyrimidin-...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK2(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784732(2-((6-(4-acetylpiperazin-1-yl)- 2-methylpyrimidin-...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784732(2-((6-(4-acetylpiperazin-1-yl)- 2-methylpyrimidin-...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784731(N-(2-chloro-6-methylphenyl)-2- ((2-methyl-6-(4- me...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784734(N-(2-chloro-6-ethoxyphenyl)-2- ((6-(4-(2- hydroxye...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetTyrosine-protein kinase ABL1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784734(N-(2-chloro-6-ethoxyphenyl)-2- ((6-(4-(2- hydroxye...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM13277(N-(2-Chloro-6-methylphenyl)-2-(6-(2-hydroxyethylam...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetTyrosine-protein kinase ABL1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM13277(N-(2-Chloro-6-methylphenyl)-2-(6-(2-hydroxyethylam...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK3(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM13277(N-(2-Chloro-6-methylphenyl)-2-(6-(2-hydroxyethylam...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784730(N-(3-fluoro-2-methoxyphenyl)-2- ((6-(4-(2- hydroxy...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM632965(US20230348453, Compound B3 | US12172993, Compound ...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetTyrosine-protein kinase ABL1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM632965(US20230348453, Compound B3 | US12172993, Compound ...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK3(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM632965(US20230348453, Compound B3 | US12172993, Compound ...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK2(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM632965(US20230348453, Compound B3 | US12172993, Compound ...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetSerine/threonine-protein kinase SIK1(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM632965(US20230348453, Compound B3 | US12172993, Compound ...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
iOmx Therapeutics

US Patent
LigandPNGBDBM784728(N-(2,6-dibromophenyl)-2- ((6-(4-(2-hydroxyethyl)pi...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/26/2026
Entry Details US Patent

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