Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 4579
TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293025BDBM293025(1-(6-{1H-pyrazolo[3,4-c]pyridin-3-yl}-2,3-dihydroi...)
Affinity DataIC50: 4.80nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293043BDBM293043(3-[1-(prop-2-enoyl)-2,3-dihydroindol-6-yl]-1H-inda...)
Affinity DataIC50: 6nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293041BDBM293041(1-(ethenesulfonyl)-6-{1H-pyrazolo[3,4-b]pyridin-3-...)
Affinity DataIC50: 7.70nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293028BDBM293028(1-[6-(6-methyl-1H-indazol-3-yl)-2,3-dihydroindol-1...)
Affinity DataKd:  7.80nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293038BDBM293038(1-[6-(1H-indazol-3-yl)-2,3-dihydroindol-1-yl]prop-...)
Affinity DataIC50: 19nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293028BDBM293028(1-[6-(6-methyl-1H-indazol-3-yl)-2,3-dihydroindol-1...)
Affinity DataIC50: 23nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293027BDBM293027(1-(6-{1H-pyrazolo[4,3-c]pyridin-3-yl}-2,3-dihydroi...)
Affinity DataIC50: 30nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293029BDBM293029((2E)-4-[6-(1H-indazol-3-yl)-2,3-dihydroindol-1-yl]...)
Affinity DataIC50: 70nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293036BDBM293036(1-[7-(6-methyl-1H-indazol-3-yl)-3,4-dihydro-2H-qui...)
Affinity DataKd:  71nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293042BDBM293042(1-(7-fluoro-6-{1H-pyrazolo[3,4-b]pyridin-3-yl}-2,3...)
Affinity DataIC50: 88nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293026BDBM293026(1-[4-(1H-indazol-3-yl)-2,3-dihydroindol-1-yl]prop-...)
Affinity DataIC50: 92nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293037BDBM293037(1-[6-(1H-indazol-3-yl)-2,3-dihydro-1,4-benzoxazin-...)
Affinity DataIC50: 140nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293036BDBM293036(1-[7-(6-methyl-1H-indazol-3-yl)-3,4-dihydro-2H-qui...)
Affinity DataIC50: 160nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293040BDBM293040(US20260015351, Compound 15-B)
Affinity DataIC50: 160nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293030BDBM293030((2E)-4-(dimethylamino)-1-[6-(1H-indazol-3-yl)-2,3-...)
Affinity DataIC50: 180nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293039BDBM293039([3,4-b]pyridin-3-yl}-2,3-dihydroindol-1-yl]prop-2-...)
Affinity DataIC50: 440nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293034BDBM293034(1-(7-{1H-pyrazolo[3,4-c]pyridin-3-yl}-3,4-dihydro-...)
Affinity DataIC50: 550nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293032BDBM293032(2-fluoro-1-[6-(1H-indazol-3-yl)-2,3-dihydroindol-1...)
Affinity DataIC50: 840nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293033BDBM293033((2E)-1-[6-(1H-indazol-3-yl)-2,3-dihydroindol-1-yl]...)
Affinity DataIC50: 1.10E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293035BDBM293035(1-(7-{1H-pyrazolo[4,3-c]pyridin-3-yl}-3,4-dihydro-...)
Affinity DataIC50: 1.40E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent

TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Axonis Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 293031BDBM293031((2E)-4-[6-(1H-indazol-3-yl)-2,3-dihydroindol-1-yl]...)
Affinity DataIC50: 3.90E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2026
Entry Details US Patent