Compile Data Set for Download or QSAR
Report error Found 218 Enz. Inhib. hit(s) with all data for entry = 12677
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793356BDBM793356((R)-4-(((3-chloro-1-(prop-2-yn-1-yl)-1H- pyrazolo[...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793353BDBM793353((4-(((3-chloro-1-(prop-2-yn-1-yl)-1H- pyrazolo[3,4...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793354BDBM793354((4-(((1-ethyl-1H-pyrazolo[3,4-b]pyridin-4- yl)amin...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793360BDBM793360(4-(((3-chloro-1-(prop-2-yn-1-yl)-1H- pyrazolo[3,4-...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793317BDBM793317(4-(((3-chloro-1-(prop-2-yn-1-yl)-1H- pyrazolo[3,4-...)
Affinity DataIC50: 10nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793316BDBM793316(4-(((3-chloro-1-(prop-2-yn-1-yl)-1H- pyrazolo[3,4-...)
Affinity DataIC50: 10nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793386BDBM793386((S)-1-ethyl-N-((1-(S- methylsulfonimidoyl)piperidi...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793357BDBM793357((S)-4-(((3-chloro-1-(prop-2-yn-1-yl)-1H- pyrazolo[...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793384BDBM793384(3-(4-(((3-chloro-1-ethyl-1H-pyrazolo[3,4-b] pyridi...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793363BDBM793363(4-(((3-chloro-1-(prop-2-yn-1-yl)-1H- pyrazolo[3,4-...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793389BDBM793389(N-(2-(4-(((3-chloro-1-ethyl-1H-pyrazolo[3,4-b] pyr...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793364BDBM793364(4-(((3-chloro-1-(cyanomethyl)-1H-pyrazolo[3,4- b]p...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793390BDBM793390(4-(((3-chloro-1-(cyanomethyl)-1H-pyrazolo[3,4- b]p...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793361BDBM793361(4-(((3-chloro-1-(cyanomethyl)-1H-pyrazolo[3,4- b]p...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793319BDBM793319((S)-4-(((1-ethyl-1H-pyrazolo[3,4-b]pyridin-4- yl)a...)
Affinity DataIC50: 10nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793318BDBM793318(N'-cyano-4-(((1-ethyl-1H-pyrazolo[3,4-b]pyridin- 4...)
Affinity DataIC50: 10nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793387BDBM793387((S)-N-((4-(((3-chloro-1-(prop-2-yn-1-yl)-1H- pyraz...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793362BDBM793362(4-(((3-chloro-1-ethyl-1H-pyrazolo[3,4-b]pyridin- 4...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793330BDBM793330(4-((3-chloro-1-ethyl-1H-pyrazolo[3,4-b]pyridin- 4-...)
Affinity DataIC50: 10nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793329BDBM793329(4-((3-chloro-1-ethyl-1H-pyrazolo[3,4-b]pyridin- 4-...)
Affinity DataIC50: 10nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793393BDBM793393(4-(((3-chloro-1-(prop-2-yn-1-yl)-1H- pyrazolo[3,4-...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793332BDBM793332((S)-(4-(((3-chloro-1-(prop-2-yn-1-yl)-1H- pyrazolo...)
Affinity DataIC50: 10nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793368BDBM793368(4-(((3-chloro-1-ethyl-1H-pyrazolo[3,4-b]pyridin- 4...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793326BDBM793326(4-((3-chloro-1-ethyl-1H-pyrazolo[3,4-b]pyridin- 4-...)
Affinity DataIC50: 10nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 3(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793391BDBM793391(4-(((3-chloro-1-(cyanomethyl)-1H-pyrazolo[3,4- b]p...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793325BDBM793325(4-((3-chloro-1-ethyl-1H-pyrazolo[3,4-b]pyridin- 4-...)
Affinity DataIC50: 10nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793391BDBM793391(4-(((3-chloro-1-(cyanomethyl)-1H-pyrazolo[3,4- b]p...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793327BDBM793327(4-((3-chloro-1-ethyl-1H-pyrazolo[3,4-b]pyridin- 4-...)
Affinity DataIC50: 10nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793392BDBM793392(4-(((3-chloro-1-ethyl-1H-pyrazolo[3,4-b]pyridin- 4...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793338BDBM793338((4-(((3-chloro-1-(prop-2-yn-1-yl)-1H- pyrazolo[3,4...)
Affinity DataIC50: 10nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 3(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793370BDBM793370(4-(((3-chloro-1-(cyanomethyl)-1H-pyrazolo[3,4- b]p...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 3(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793395BDBM793395((R)-4-(((3-chloro-1-(cyanomethyl)-1H- pyrazolo[3,4...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793337BDBM793337((S)-(4-(((3-chloro-1-(prop-2-yn-1-yl)-1H- pyrazolo...)
Affinity DataIC50: 10nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793370BDBM793370(4-(((3-chloro-1-(cyanomethyl)-1H-pyrazolo[3,4- b]p...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793395BDBM793395((R)-4-(((3-chloro-1-(cyanomethyl)-1H- pyrazolo[3,4...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793340BDBM793340(2-(3-chloro-4-((4-(S- methylsulfonimidoyl)benzyl)a...)
Affinity DataIC50: 10nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 793334BDBM793334(2-(3-chloro-4-((4-(S-methylsulfonimidoyl) benzyl)o...)
Affinity DataIC50: 10nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 3(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793394BDBM793394((S)-4-(((3-chloro-1-(cyanomethyl)-1H- pyrazolo[3,4...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793369BDBM793369(N'-cyano-4-(((1-ethyl-1H-pyrazolo[3,4- b]pyridin-4...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793394BDBM793394((S)-4-(((3-chloro-1-(cyanomethyl)-1H- pyrazolo[3,4...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793336BDBM793336((R)-(4-(((3-chloro-1-(prop-2-yn-1-yl)-1H- pyrazolo...)
Affinity DataIC50: 10nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 793335BDBM793335((4-(((3-chloro-1-(prop-2-yn-1-yl)-1H-pyrazolo [3,4...)
Affinity DataIC50: 10nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 3(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793372BDBM793372((R)-4-(((3-chloro-1-(prop-2-yn-1-yl)-1H- pyrazolo[...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 793372BDBM793372((R)-4-(((3-chloro-1-(prop-2-yn-1-yl)-1H- pyrazolo[...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793397BDBM793397((R)-4-(((3-chloro-1-(cyanomethyl)-1H- pyrazolo[3,4...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793344BDBM793344((4-(((3-chloro-1-ethyl-1H-pyrazolo[3,4-b] pyridin-...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793342BDBM793342((R)-2-(3-chloro-4-((4-(S- methylsulfonimidoyl)benz...)
Affinity DataIC50: 10nMAssay Description:AlphaScreen (Amplified Luminescent Proximity Homogeneous Assay, ALPHA, Perkin Elmer) is a non-radioactive bead-based proximity assay technology to st...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 3(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793371BDBM793371(4-(((3-chloro-1-(prop-2-yn-1-yl)-1H- pyrazolo[3,4-...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793371BDBM793371(4-(((3-chloro-1-(prop-2-yn-1-yl)-1H- pyrazolo[3,4-...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Gossamer Bio Services

US Patent
LigandChemical structure of BindingDB Monomer ID 793396BDBM793396((S)-4-(((3-chloro-1-(cyanomethyl)-1H- pyrazolo[3,4...)
Affinity DataIC50: 10nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/1/2026
Entry Details
US Patent

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