Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 13443
TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793854BDBM793854(US20260055104, Compound I)
Affinity DataIC50: 0.670nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/9/2026
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 2 (PARP2)(Human)
Haisco Pharmaceutical Group Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793854BDBM793854(US20260055104, Compound I)
Affinity DataIC50: 27.5nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/9/2026
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-2 (PARP5B)(Human)
Haisco Pharmaceutical Group Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793854BDBM793854(US20260055104, Compound I)
Affinity DataIC50: 576nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/9/2026
Entry Details
US Patent

TargetProtein mono-ADP-ribosyltransferase PARP15(Human)
Haisco Pharmaceutical Group Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793854BDBM793854(US20260055104, Compound I)
Affinity DataIC50: 4.30E+3nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/9/2026
Entry Details
US Patent

TargetProtein mono-ADP-ribosyltransferase TIPARP (PARP7)(Human)
Haisco Pharmaceutical Group Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793854BDBM793854(US20260055104, Compound I)
Affinity DataIC50: 5.36E+3nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/9/2026
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1 (PARP5A)(Human)
Haisco Pharmaceutical Group Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793854BDBM793854(US20260055104, Compound I)
Affinity DataIC50: 6.08E+3nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/9/2026
Entry Details
US Patent

TargetProtein mono-ADP-ribosyltransferase PARP6(Human)
Haisco Pharmaceutical Group Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793854BDBM793854(US20260055104, Compound I)
Affinity DataIC50: 6.86E+3nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/9/2026
Entry Details
US Patent

TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
Haisco Pharmaceutical Group Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793854BDBM793854(US20260055104, Compound I)
Affinity DataIC50: 7.06E+3nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/9/2026
Entry Details
US Patent