Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 5888
LigandChemical structure of BindingDB Monomer ID 98618BDBM98618(US8470847, 81 | 2-amino-1-ethyl-7-[3-hydroxy-3-(3-...)
Affinity DataIC50: 2nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 98616BDBM98616(2-amino-1-cyclohexyl-7-(3-hydroxy-4-methoxy-3-meth...)
Affinity DataIC50: 5nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 98610BDBM98610(2-amino-1-ethyl-7-[3-hydroxy-3-(3-methoxyphenyl)bu...)
Affinity DataIC50: 6nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 98615BDBM98615(2-amino-1-ethyl-7-(3-hydroxy-3-phenyl-but-1-ynyl)-...)
Affinity DataIC50: 14nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 98608BDBM98608(2-amino-1-ethyl-7-[2-(1-hydroxycyclobutyl)ethynyl]...)
Affinity DataIC50: 21nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 98617BDBM98617(2-amino-1-ethyl-7-(3-hydroxy-4-methoxy-3-methyl-bu...)
Affinity DataIC50: 23nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 98605BDBM98605(2-amino-1-ethyl-7-[2-(3-hydroxytetrahydrofuran-3-y...)
Affinity DataIC50: 23nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 98611BDBM98611(2-amino-7-(3,4-dihydroxy-3-methyl-but-1-ynyl)-N-me...)
Affinity DataIC50: 34nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 98607BDBM98607(2-amino-7-(3-cyclopropyl-3-hydroxy-prop-1-ynyl)-1-...)
Affinity DataIC50: 37nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 98618BDBM98618(US8470847, 81 | 2-amino-1-ethyl-7-[3-hydroxy-3-(3-...)
Affinity DataIC50: 38nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 98612BDBM98612(2-amino-7-(3-hydroxy-3-methyl-but-1-ynyl)-N-methyl...)
Affinity DataIC50: 40nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 98614BDBM98614(2-amino-7-(3,4-dihydroxy-3-methyl-but-1-ynyl)-1-et...)
Affinity DataIC50: 43nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 98606BDBM98606(2-amino-7-(3,4-dihydroxy-3-methyl-but-1-ynyl)-1-et...)
Affinity DataIC50: 46nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 98613BDBM98613(2-amino-7-(3-hydroxy-4-methoxy-3-methyl-but-1-ynyl...)
Affinity DataIC50: 65nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 98609BDBM98609(2-amino-7-(3-hydroxy-4-methoxy-3-methyl-but-1-ynyl...)
Affinity DataIC50: 257nMT: 2°CAssay Description:Activity of VEGFR-3 is measured by ELISA assay by measuring the intensity of phosphorylation of the substrate poly Glu-Tyr.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
US Patent