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Found 211 Enz. Inhib. hit(s) with all data for entry = 5920
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100437(US8501732, I-1)
Affinity DataIC50:  1nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100549(US8501732, I-109)
Affinity DataIC50:  4nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100445(US8501732, I-9)
Affinity DataIC50:  4nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100609(US8501732, I-169)
Affinity DataIC50:  4nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100550(US8501732, I-110)
Affinity DataIC50:  4nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100551(US8501732, I-111)
Affinity DataIC50:  5nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100573(US8501732, I-133)
Affinity DataIC50:  6nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100552(US8501732, I-112)
Affinity DataIC50:  6nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100553(US8501732, I-113)
Affinity DataIC50:  7nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100554(US8501732, I-114)
Affinity DataIC50:  7nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100448(US8501732, I-12)
Affinity DataIC50:  7nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100438(US8501732, I-2)
Affinity DataIC50:  7nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100574(US8501732, I-134)
Affinity DataIC50:  7nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100555(US8501732, I-115)
Affinity DataIC50:  8nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100575(US8501732, I-135)
Affinity DataIC50:  8nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100556(US8501732, I-116)
Affinity DataIC50:  8nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100439(US8501732, I-3)
Affinity DataIC50:  9nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100610(US8501732, I-170)
Affinity DataIC50:  10nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100557(US8501732, I-117)
Affinity DataIC50:  10nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100502(US8501732, I-62)
Affinity DataIC50:  11nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100558(US8501732, I-118)
Affinity DataIC50:  11nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100576(US8501732, I-136)
Affinity DataIC50:  12nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100590(US8501732, I-150)
Affinity DataIC50:  12nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100577(US8501732, I-137)
Affinity DataIC50:  12nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100559(US8501732, I-119)
Affinity DataIC50:  13nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100469(US8501732, I-29)
Affinity DataIC50:  13nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100579(US8501732, I-139)
Affinity DataIC50:  13nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100578(US8501732, I-138)
Affinity DataIC50:  13nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100580(US8501732, I-140)
Affinity DataIC50:  14nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100443(US8501732, I-7)
Affinity DataIC50:  14nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100440(US8501732, I-4)
Affinity DataIC50:  14nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100560(US8501732, I-120)
Affinity DataIC50:  15nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100561(US8501732, I-121)
Affinity DataIC50:  15nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100581(US8501732, I-141)
Affinity DataIC50:  15nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100572(US8501732, I-132)
Affinity DataIC50:  15nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100562(US8501732, I-122)
Affinity DataIC50:  15nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100531(US8501732, I-91)
Affinity DataIC50:  16nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100563(US8501732, I-123)
Affinity DataIC50:  16nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100564(US8501732, I-124)
Affinity DataIC50:  17nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100503(US8501732, I-63)
Affinity DataIC50:  17nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100582(US8501732, I-142)
Affinity DataIC50:  17nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100592(US8501732, I-152)
Affinity DataIC50:  18nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100504(US8501732, I-64)
Affinity DataIC50:  18nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100470(US8501732, I-30)
Affinity DataIC50:  18nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100506(US8501732, I-66)
Affinity DataIC50:  19nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100505(US8501732, I-65)
Affinity DataIC50:  19nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100507(US8501732, I-67)
Affinity DataIC50:  20nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100532(US8501732, I-92)
Affinity DataIC50:  21nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100508(US8501732, I-68)
Affinity DataIC50:  21nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100565(US8501732, I-125)
Affinity DataIC50:  22nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
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