Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 5951
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Sanofi

US Patent
LigandPNGBDBM102430(US8536173, 5)
Affinity DataIC50: 11nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2013
Entry Details
US Patent

Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Sanofi

US Patent
LigandPNGBDBM102428(US8536173, 3)
Affinity DataIC50: 21nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2013
Entry Details
US Patent

Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Sanofi

US Patent
LigandPNGBDBM102429(US8536173, 4)
Affinity DataIC50: 23nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2013
Entry Details
US Patent

Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Sanofi

US Patent
LigandPNGBDBM102434(US8536173, 9)
Affinity DataIC50: 31nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2013
Entry Details
US Patent

Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Sanofi

US Patent
LigandPNGBDBM102427(US8536173, 2)
Affinity DataIC50: 32nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2013
Entry Details
US Patent

Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Sanofi

US Patent
LigandPNGBDBM102432(US8536173, 7)
Affinity DataIC50: 45nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2013
Entry Details
US Patent

Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Sanofi

US Patent
LigandPNGBDBM102431(US8536173, 6)
Affinity DataIC50: 57nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2013
Entry Details
US Patent

Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Sanofi

US Patent
LigandPNGBDBM102426(US8536173, 1)
Affinity DataIC50: 68nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2013
Entry Details
US Patent

Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Sanofi

US Patent
LigandPNGBDBM102433(US8536173, 8)
Affinity DataIC50: 204nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2013
Entry Details
US Patent

Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Sanofi

US Patent
LigandPNGBDBM8528(US8536173, 10)
Affinity DataIC50: 720nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2013
Entry Details
US Patent