Compile Data Set for Download or QSAR
maximum 50k data
Found 17 Enz. Inhib. hit(s) with all data for entry = 5988
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101038(US8524917, 11 | US8563594, 169)
Affinity DataIC50:  5nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101039(US8524917, 12 | US8563594, 170)
Affinity DataIC50:  6nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM103621(US8563594, 171)
Affinity DataIC50:  17nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101037(US8524917, 10 | US8563594, 168)
Affinity DataIC50:  19nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM103616(US8563594, 166)
Affinity DataIC50:  31nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM103614(US8563594, 164)
Affinity DataIC50:  35nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM103617(US8563594, 167)
Affinity DataIC50:  209nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM103604(US8563594, 153)
Affinity DataIC50:  231nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM103611(US8563594, 160)
Affinity DataIC50:  319nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM38239(US8563594, 154 | US8563594, Unnumbered 2)
Affinity DataIC50:  319nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM38239(US8563594, 154 | US8563594, Unnumbered 2)
Affinity DataIC50:  319nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM103608(US8563594, 157)
Affinity DataIC50:  1.10E+3nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM103603(US8563594, 152)
Affinity DataIC50:  1.60E+3nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM103609(US8563594, 158)
Affinity DataIC50:  1.80E+3nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM103606(US8563594, 155)
Affinity DataIC50:  1.80E+3nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM103613(US8563594, 162)
Affinity DataIC50:  1.90E+3nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM103612(US8563594, 161)
Affinity DataIC50:  4.00E+3nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent