Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 6353
TargetSomatostatin receptor type 3(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM124131(US8754099, 22)
Affinity DataIC50: 1.20nMpH: 7.8 T: 2°CAssay Description:The receptor-ligand binding Scintillation Proximity Assay (SPA) (N. D. Cook. Drug Discovery Today 1 (1996), pp. 287-294) for SSTR3 was performed with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetSomatostatin receptor type 3(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM124130(US8754099, 21)
Affinity DataIC50: 1.70nMpH: 7.8 T: 2°CAssay Description:The receptor-ligand binding Scintillation Proximity Assay (SPA) (N. D. Cook. Drug Discovery Today 1 (1996), pp. 287-294) for SSTR3 was performed with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetSomatostatin receptor type 3(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM124114(US8754099, 4)
Affinity DataIC50: 2.60nMpH: 7.8 T: 2°CAssay Description:The receptor-ligand binding Scintillation Proximity Assay (SPA) (N. D. Cook. Drug Discovery Today 1 (1996), pp. 287-294) for SSTR3 was performed with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetSomatostatin receptor type 3(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM124129(US8754099, 20)
Affinity DataIC50: 4.60nMpH: 7.8 T: 2°CAssay Description:The receptor-ligand binding Scintillation Proximity Assay (SPA) (N. D. Cook. Drug Discovery Today 1 (1996), pp. 287-294) for SSTR3 was performed with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent

TargetSomatostatin receptor type 3(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM124113(US8754099, 3)
Affinity DataIC50: 43.8nMpH: 7.8 T: 2°CAssay Description:The receptor-ligand binding Scintillation Proximity Assay (SPA) (N. D. Cook. Drug Discovery Today 1 (1996), pp. 287-294) for SSTR3 was performed with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2014
Entry Details
US Patent