Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 6430
TargetFatty acid synthase(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 128366BDBM128366(US8802864, 132)
Affinity DataIC50: 3nMpH: 7.0Assay Description:Assay #1:Inhibition of FAS activity can be measured based on the detection of residual NADPH substrate after the FAS assay is quenched. This assay is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetFatty acid synthase(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 128362BDBM128362(US8802864, 42)
Affinity DataIC50: 5nMpH: 7.0Assay Description:Assay #1:Inhibition of FAS activity can be measured based on the detection of residual NADPH substrate after the FAS assay is quenched. This assay is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetFatty acid synthase(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 128359BDBM128359(US8802864, 14)
Affinity DataIC50: 6nMpH: 7.0Assay Description:Assay #1:Inhibition of FAS activity can be measured based on the detection of residual NADPH substrate after the FAS assay is quenched. This assay is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetFatty acid synthase(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 119133BDBM119133((S)-4-(4-(Benzofuran-5-yl)phenyl)-3-((1-(cycloprop...)
Affinity DataIC50: 10nMpH: 7.0Assay Description:Assay #1:Inhibition of FAS activity can be measured based on the detection of residual NADPH substrate after the FAS assay is quenched. This assay is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetFatty acid synthase(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 128360BDBM128360(US8802864, 23)
Affinity DataIC50: 13nMpH: 7.0Assay Description:Assay #1:Inhibition of FAS activity can be measured based on the detection of residual NADPH substrate after the FAS assay is quenched. This assay is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetFatty acid synthase(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 128363BDBM128363(US8802864, 67)
Affinity DataIC50: 16nMpH: 7.0Assay Description:Assay #1:Inhibition of FAS activity can be measured based on the detection of residual NADPH substrate after the FAS assay is quenched. This assay is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetFatty acid synthase(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 128358BDBM128358(US8802864, 7)
Affinity DataIC50: 20nMpH: 7.0Assay Description:Assay #1:Inhibition of FAS activity can be measured based on the detection of residual NADPH substrate after the FAS assay is quenched. This assay is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetFatty acid synthase(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 128365BDBM128365(US8802864, 116)
Affinity DataIC50: 40nMpH: 7.0Assay Description:Assay #1:Inhibition of FAS activity can be measured based on the detection of residual NADPH substrate after the FAS assay is quenched. This assay is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetFatty acid synthase(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 128357BDBM128357(US8802864, 4)
Affinity DataIC50: 126nMpH: 7.0Assay Description:Assay #1:Inhibition of FAS activity can be measured based on the detection of residual NADPH substrate after the FAS assay is quenched. This assay is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetFatty acid synthase(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 128361BDBM128361(US8802864, 38)
Affinity DataIC50: 158nMpH: 7.0Assay Description:Assay #1:Inhibition of FAS activity can be measured based on the detection of residual NADPH substrate after the FAS assay is quenched. This assay is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetFatty acid synthase(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 128364BDBM128364(US8802864, 95)
Affinity DataIC50: 200nMpH: 7.0Assay Description:Assay #1:Inhibition of FAS activity can be measured based on the detection of residual NADPH substrate after the FAS assay is quenched. This assay is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetFatty acid synthase(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 128367BDBM128367(US8802864, 158)
Affinity DataIC50: 398nMpH: 7.0Assay Description:Assay #1:Inhibition of FAS activity can be measured based on the detection of residual NADPH substrate after the FAS assay is quenched. This assay is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent