Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 6528
TargetRegulator of G-protein signaling 4(Homo sapiens (Human))
University of Michigan

US Patent
LigandPNGBDBM50384774(CHEMBL1917204 | US20230414581, Compound 6)
Affinity DataIC50:  30nMAssay Description:FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRegulator of G-protein signaling 19(Homo sapiens (Human))
University of Michigan

US Patent
LigandPNGBDBM50384774(CHEMBL1917204 | US20230414581, Compound 6)
Affinity DataIC50:  120nMAssay Description:FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRegulator of G-protein signaling 16(Homo sapiens (Human))
University of Michigan

US Patent
LigandPNGBDBM50384774(CHEMBL1917204 | US20230414581, Compound 6)
Affinity DataIC50:  3.50E+3nMAssay Description:FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
University of Michigan

US Patent
LigandPNGBDBM50384774(CHEMBL1917204 | US20230414581, Compound 6)
Affinity DataIC50:  1.10E+4nMAssay Description:FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRegulator of G-protein signaling 4(Homo sapiens (Human))
University of Michigan

US Patent
LigandPNGBDBM136369(US8865750, CCG- 203780)
Affinity DataIC50:  3.20E+4nMAssay Description:FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRegulator of G-protein signaling 4(Homo sapiens (Human))
University of Michigan

US Patent
LigandPNGBDBM50384773(CHEMBL2037371)
Affinity DataIC50:  9.30E+4nMAssay Description:FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
University of Michigan

US Patent
LigandPNGBDBM50384773(CHEMBL2037371)
Affinity DataIC50: >1.00E+5nMAssay Description:FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
University of Michigan

US Patent
LigandPNGBDBM136368(US8865750, CCG- 203778)
Affinity DataIC50: >1.00E+5nMAssay Description:FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
University of Michigan

US Patent
LigandPNGBDBM136369(US8865750, CCG- 203780)
Affinity DataIC50: >1.00E+5nMAssay Description:FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRegulator of G-protein signaling 4(Homo sapiens (Human))
University of Michigan

US Patent
LigandPNGBDBM136368(US8865750, CCG- 203778)
Affinity DataIC50: >1.00E+5nMAssay Description:FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent