Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 6599
TargetEpidermal growth factor receptor(Human)
Qilu Pharmaceutical

US Patent
LigandPNGBDBM140984(US8916574, Compound 1)
Affinity DataIC50: 2.71nMT: 2°CAssay Description:In vitro kinase analysis was performed by using HTScan EGF Receptor Kinase Assay Kit (#7909) and HTScan HER2/ErbB2 Kinase Assay Kit (#7058) from Cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2015
Entry Details
US Patent

TargetEpidermal growth factor receptor(Human)
Qilu Pharmaceutical

US Patent
LigandPNGBDBM140988(US8916574, Compound 5)
Affinity DataIC50: 14.6nMT: 2°CAssay Description:In vitro kinase analysis was performed by using HTScan EGF Receptor Kinase Assay Kit (#7909) and HTScan HER2/ErbB2 Kinase Assay Kit (#7058) from Cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2015
Entry Details
US Patent

TargetEpidermal growth factor receptor(Human)
Qilu Pharmaceutical

US Patent
LigandPNGBDBM140987(US8916574, Compound 4)
Affinity DataIC50: 15.5nMT: 2°CAssay Description:In vitro kinase analysis was performed by using HTScan EGF Receptor Kinase Assay Kit (#7909) and HTScan HER2/ErbB2 Kinase Assay Kit (#7058) from Cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/11/2015
Entry Details
US Patent

TargetEpidermal growth factor receptor(Human)
Qilu Pharmaceutical

US Patent
LigandPNGBDBM140989(US8916574, Compound 6)
Affinity DataIC50: 32.4nMT: 2°CAssay Description:In vitro kinase analysis was performed by using HTScan EGF Receptor Kinase Assay Kit (#7909) and HTScan HER2/ErbB2 Kinase Assay Kit (#7058) from Cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2015
Entry Details
US Patent

TargetEpidermal growth factor receptor(Human)
Qilu Pharmaceutical

US Patent
LigandPNGBDBM140985(US8916574, Compound 2)
Affinity DataIC50: 52.7nMT: 2°CAssay Description:In vitro kinase analysis was performed by using HTScan EGF Receptor Kinase Assay Kit (#7909) and HTScan HER2/ErbB2 Kinase Assay Kit (#7058) from Cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2015
Entry Details
US Patent

TargetEpidermal growth factor receptor(Human)
Qilu Pharmaceutical

US Patent
LigandPNGBDBM140986(US8916574, Compound 3)
Affinity DataIC50: 56.2nMT: 2°CAssay Description:In vitro kinase analysis was performed by using HTScan EGF Receptor Kinase Assay Kit (#7909) and HTScan HER2/ErbB2 Kinase Assay Kit (#7058) from Cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2015
Entry Details
US Patent