Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 6875
TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM155363(US9006269, 9 | US10383871, Example 9 | US10918640,...)
Affinity DataIC50: 3nMpH: 8.2 T: 2°CAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM155368(US9006269, 15 | US10383871, Example 15 | US1091864...)
Affinity DataIC50: 7nMpH: 8.2 T: 2°CAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM155359(US9006269, 5 | US10383871, Example 5 | US10918640,...)
Affinity DataIC50: 9nMpH: 8.2 T: 2°CAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM155372(US9006269, 17 | US10383871, Example 17 | US1091864...)
Affinity DataIC50: 12nMpH: 8.2 T: 2°CAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM155366(US9006269, 12 | US10383871, Example 12 | US1091864...)
Affinity DataIC50: 12nMpH: 8.2 T: 2°CAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM155370(US9006269, 14)
Affinity DataIC50: 14nMpH: 8.2 T: 2°CAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM155373(US9006269, 18 | US10383871, Example 18)
Affinity DataIC50: 16nMpH: 8.2 T: 2°CAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM155362(US9006269, 8 | US10383871, Example 8 | US10918640,...)
Affinity DataIC50: 18nMpH: 8.2 T: 2°CAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM155361(US9006269, 7 | US10383871, Example 7 | US10918640,...)
Affinity DataIC50: 19nMpH: 8.2 T: 2°CAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM155365(US9006269, 11 | US10383871, Example 11 | US1091864...)
Affinity DataIC50: 19nMpH: 8.2 T: 2°CAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM155369(US9006269, 19 | US10383871, Example 19 | US1091864...)
Affinity DataIC50: 26nMpH: 8.2 T: 2°CAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM155367(US9006269, 13 | US10383871, Example 13 | US1091864...)
Affinity DataIC50: 38nMpH: 8.2 T: 2°CAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM155371(US9006269, 16 | US10383871, Example 16 | US1091864...)
Affinity DataIC50: 42nMpH: 8.2 T: 2°CAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM155364(US9006269, 10 | US10383871, Example 10 | US1091864...)
Affinity DataIC50: 49nMpH: 8.2 T: 2°CAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Vernalis (R&D)

US Patent
LigandPNGBDBM155358(US9006269, 4 | US10383871, Example 4 | US10918640,...)
Affinity DataIC50: 67nMpH: 8.2 T: 2°CAssay Description:FAAH activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolysis of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM155360(US9006269, 6 | US10383871, Example 6 | US10918640,...)
Affinity DataIC50: 73nMpH: 8.2 T: 2°CAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Vernalis (R&D)

US Patent
LigandPNGBDBM155357(US9006269, 3 | US10383871, Example 3 | US10918640,...)
Affinity DataIC50: 77nMpH: 8.2 T: 2°CAssay Description:FAAH activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolysis of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Vernalis (R&D)

US Patent
LigandPNGBDBM155355(US9006269, 1 | US10383871, Example 1 | US10918640,...)
Affinity DataIC50: 135nMpH: 8.2 T: 2°CAssay Description:FAAH activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolysis of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Vernalis (R&D)

US Patent
LigandPNGBDBM155356(US9006269, 2 | US10383871, Example 2 | US10918640,...)
Affinity DataIC50: 279nMpH: 8.2 T: 2°CAssay Description:FAAH activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolysis of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent