Compile Data Set for Download or QSAR
maximum 50k data
Found 44 Enz. Inhib. hit(s) with all data for entry = 6916
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159297(US9034897, 14a)
Affinity DataIC50:  70nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159298(US9034897, 14b)
Affinity DataIC50:  83.1nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159259(US9034897, 11a)
Affinity DataIC50:  171nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159321(US9034897, 22a)
Affinity DataIC50:  180nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159260(US9034897, 11b)
Affinity DataIC50:  190nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159261(US9034897, 11c)
Affinity DataIC50:  204nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159262(US9034897, 11d)
Affinity DataIC50:  226nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159315(US9034897, 19a)
Affinity DataIC50:  231nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159263(US9034897, 11e)
Affinity DataIC50:  239nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159299(US9034897, 14c)
Affinity DataIC50:  250nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159306(US9034897, 17a)
Affinity DataIC50:  260nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159264(US9034897, 11f)
Affinity DataIC50:  270nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159265(US9034897, 11g)
Affinity DataIC50:  350nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159266(US9034897, 11h)
Affinity DataIC50:  370nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159267(US9034897, 11i)
Affinity DataIC50:  375nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159318(US9034897, 21a)
Affinity DataIC50:  393nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159268(US9034897, 11j)
Affinity DataIC50:  439nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159269(US9034897, 11k)
Affinity DataIC50:  442nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159304(US9034897, 16a)
Affinity DataIC50:  446nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159291(US9034897, 12b)
Affinity DataIC50:  479nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM47354(US9034897, 11l)
Affinity DataIC50:  495nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159317(US9034897, 20a)
Affinity DataIC50:  500nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159307(US9034897, 18a)
Affinity DataIC50:  500nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM47355(US9034897, 11m)
Affinity DataIC50:  518nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM47356(US9034897, 11n)
Affinity DataIC50:  568nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM47357(US9034897, 11o)
Affinity DataIC50:  675nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159274(US9034897, 11p)
Affinity DataIC50:  685nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159290(US9034897, 12a)
Affinity DataIC50:  712nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159275(US9034897, 11q)
Affinity DataIC50:  773nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159276(US9034897, 11r)
Affinity DataIC50:  789nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159277(US9034897, 11s)
Affinity DataIC50:  804nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159278(US9034897, 11t)
Affinity DataIC50:  881nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159279(US9034897, 11u)
Affinity DataIC50:  1.01E+3nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159305(US9034897, 16b)
Affinity DataIC50:  1.16E+3nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159280(US9034897, 11v)
Affinity DataIC50:  1.19E+3nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159281(US9034897, 11w)
Affinity DataIC50:  1.26E+3nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159282(US9034897, 11x)
Affinity DataIC50:  1.52E+3nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159283(US9034897, 11y)
Affinity DataIC50:  1.92E+3nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159284(US9034897, 11z)
Affinity DataIC50:  2.13E+3nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM47359(US9034897, 11aa)
Affinity DataIC50:  2.22E+3nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM47360(US9034897, 11ab)
Affinity DataIC50:  2.97E+3nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM47361(US9034897, 11ac)
Affinity DataIC50:  3.88E+3nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM47362(US9034897, 11ad)
Affinity DataIC50:  6.89E+3nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM159308(US9034897, 18b)
Affinity DataIC50:  8.19E+3nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In DepthDetails US Patent