Compile Data Set for Download or QSAR
Report error Found 47 Enz. Inhib. hit(s) with all data for entry = 6931
TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160301(US9040691, 29)
Affinity DataIC50: 1nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160276(US9040691, 4)
Affinity DataIC50: 1nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160312(US9040691, 42 | US9040691, 41 | US9040691, 40)
Affinity DataIC50: 1.20nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160277(US9040691, 5)
Affinity DataIC50: 1.30nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160283(US9040691, 11)
Affinity DataIC50: 1.90nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160315(US9040691, 43)
Affinity DataIC50: 1.90nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160302(US9040691, 30)
Affinity DataIC50: 2nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160279(US9040691, 7)
Affinity DataIC50: 2nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160273(US9040691, 1)
Affinity DataIC50: 2nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160289(US9040691, 17)
Affinity DataIC50: 2nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160288(US9040691, 16)
Affinity DataIC50: 2.60nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160274(US9040691, 2)
Affinity DataIC50: 2.80nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160309(US9040691, 37)
Affinity DataIC50: 3nMAssay Description:ALKl (Invitrogen, Carlsbad, CA, USA) kinase activity was measured at ProQinase GmbH ( Freiburg. Germany) in a radiometric assay using gamma-33P-ATP a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160283(US9040691, 11)
Affinity DataIC50: 3nMAssay Description:ALKl (Invitrogen, Carlsbad, CA, USA) kinase activity was measured at ProQinase GmbH ( Freiburg. Germany) in a radiometric assay using gamma-33P-ATP a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160312(US9040691, 42 | US9040691, 41 | US9040691, 40)
Affinity DataIC50: 3.20nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160312(US9040691, 42 | US9040691, 41 | US9040691, 40)
Affinity DataIC50: 3.5nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160316(US9040691, 44)
Affinity DataIC50: 3.80nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160310(US9040691, 38)
Affinity DataIC50: 4nMAssay Description:ALKl (Invitrogen, Carlsbad, CA, USA) kinase activity was measured at ProQinase GmbH ( Freiburg. Germany) in a radiometric assay using gamma-33P-ATP a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160285(US9040691, 13)
Affinity DataIC50: 4nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160303(US9040691, 31)
Affinity DataIC50: 4nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160304(US9040691, 32)
Affinity DataIC50: 4nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160275(US9040691, 3)
Affinity DataIC50: 4nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160306(US9040691, 34)
Affinity DataIC50: 4.10nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160280(US9040691, 36 | US9040691, 35 | US9040691, 8)
Affinity DataIC50: 4.40nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160286(US9040691, 14)
Affinity DataIC50: 5.30nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160311(US9040691, 39)
Affinity DataIC50: 5.70nMAssay Description:ALKl (Invitrogen, Carlsbad, CA, USA) kinase activity was measured at ProQinase GmbH ( Freiburg. Germany) in a radiometric assay using gamma-33P-ATP a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160281(US9040691, 9)
Affinity DataIC50: 5.70nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160284(US9040691, 12)
Affinity DataIC50: 5.90nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160279(US9040691, 7)
Affinity DataIC50: 6.70nMAssay Description:ALKl (Invitrogen, Carlsbad, CA, USA) kinase activity was measured at ProQinase GmbH ( Freiburg. Germany) in a radiometric assay using gamma-33P-ATP a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160280(US9040691, 36 | US9040691, 35 | US9040691, 8)
Affinity DataIC50: 6.90nMAssay Description:ALKl (Invitrogen, Carlsbad, CA, USA) kinase activity was measured at ProQinase GmbH ( Freiburg. Germany) in a radiometric assay using gamma-33P-ATP a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160282(US9040691, 10)
Affinity DataIC50: 8nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160305(US9040691, 33)
Affinity DataIC50: 15nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160294(US9040691, 22)
Affinity DataIC50: 17nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160291(US9040691, 19)
Affinity DataIC50: 19nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160280(US9040691, 36 | US9040691, 35 | US9040691, 8)
Affinity DataIC50: 21nMAssay Description:ALKl (Invitrogen, Carlsbad, CA, USA) kinase activity was measured at ProQinase GmbH ( Freiburg. Germany) in a radiometric assay using gamma-33P-ATP a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM51425(US9040691, 21)
Affinity DataIC50: 25nMAssay Description:ALKl (Invitrogen, Carlsbad, CA, USA) kinase activity was measured at ProQinase GmbH ( Freiburg. Germany) in a radiometric assay using gamma-33P-ATP a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160298(US9040691, 26)
Affinity DataIC50: 30nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160292(US9040691, 20)
Affinity DataIC50: 30nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160295(US9040691, 23)
Affinity DataIC50: 30nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160278(US9040691, 6)
Affinity DataIC50: 40nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160287(US9040691, 15)
Affinity DataIC50: 60nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160297(US9040691, 25)
Affinity DataIC50: 65nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160299(US9040691, 27)
Affinity DataIC50: 70nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160290(US9040691, 18)
Affinity DataIC50: 80nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160300(US9040691, 28)
Affinity DataIC50: 124nMAssay Description:ALKl (Invitrogen, Carlsbad, CA, USA) kinase activity was measured at ProQinase GmbH ( Freiburg. Germany) in a radiometric assay using gamma-33P-ATP a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160296(US9040691, 24)
Affinity DataIC50: 140nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSerine/threonine-protein kinase receptor R3(Human)
Bayer Intellectual Property

US Patent
LigandPNGBDBM160300(US9040691, 28)
Affinity DataIC50: 170nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent