Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 6932
TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM160321(US9040693, 22)
Affinity DataIC50: 2nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM160326(US9040693, 146)
Affinity DataIC50: 10nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM160329(US9040693, 233)
Affinity DataIC50: 15nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM160330(US9040693, 367)
Affinity DataIC50: 15nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM160327(US9040693, 191)
Affinity DataIC50: 17nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM160325(US9040693, 95)
Affinity DataIC50: 19nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM160328(US9040693, 202)
Affinity DataIC50: 20nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM160332(US9040693, 420)
Affinity DataIC50: 29nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM160324(US9040693, 48)
Affinity DataIC50: 29nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM160331(US9040693, 414)
Affinity DataIC50: 42nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM160319(US9040693, 3)
Affinity DataIC50: 80nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM160322(US9040693, 25)
Affinity DataIC50: 85nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM160320(US9040693, 17)
Affinity DataIC50: 101nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM160318(US9040693, 2)
Affinity DataIC50: 199nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetGonadotropin-releasing hormone receptor(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM160323(US9040693, 31)
Affinity DataIC50: 272nMT: 2°CAssay Description:Antagonizing effect of compounds for human GnRHR1 was evaluated by change of calcium levels in GnRH-stimulated cells. After removing the culture medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent