Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 7284
TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186202BDBM186202(US9163013, 19)
Affinity DataIC50: 10nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186195BDBM186195(US9163013, 12)
Affinity DataIC50: 10nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186204BDBM186204(US9163013, 21)
Affinity DataIC50: 10nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186200BDBM186200(US9163013, 17)
Affinity DataIC50: 20nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186203BDBM186203(US9163013, 20)
Affinity DataIC50: 20nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186190BDBM186190(US9163013, 7)
Affinity DataIC50: 130nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186191BDBM186191(US9163013, 8)
Affinity DataIC50: 170nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186192BDBM186192(US9163013, 9)
Affinity DataIC50: 210nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186205BDBM186205(US9163013, 22)
Affinity DataIC50: 210nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186197BDBM186197(US9163013, 14)
Affinity DataIC50: 230nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186198BDBM186198(US9163013, 15)
Affinity DataIC50: 260nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186201BDBM186201(US9163013, 18)
Affinity DataIC50: 300nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186186BDBM186186(US9163013, 3)
Affinity DataIC50: 310nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186213BDBM186213(US9163013, 30)
Affinity DataIC50: 310nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186193BDBM186193(US9163013, 10)
Affinity DataIC50: 310nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186210BDBM186210(US9163013, 27)
Affinity DataIC50: 310nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186212BDBM186212(US9163013, 29)
Affinity DataIC50: 320nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186206BDBM186206(US9163013, 23)
Affinity DataIC50: 330nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186184BDBM186184(US9163013, 1)
Affinity DataIC50: 350nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186188BDBM186188(US9163013, 5)
Affinity DataIC50: 350nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186199BDBM186199(US9163013, 16)
Affinity DataIC50: 360nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186194BDBM186194(US9163013, 11)
Affinity DataIC50: 360nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186189BDBM186189(US9163013, 6)
Affinity DataIC50: 400nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186207BDBM186207(US9163013, 24)
Affinity DataIC50: 400nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186211BDBM186211(US9163013, 28)
Affinity DataIC50: 450nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186185BDBM186185(US9163013, 2)
Affinity DataIC50: 560nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186187BDBM186187(US9163013, 4)
Affinity DataIC50: 640nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186196BDBM186196(US9163013, 13)
Affinity DataIC50: 950nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186208BDBM186208(US9163013, 25)
Affinity DataIC50: 1.40E+3nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetCyclin-dependent kinase 16(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186184BDBM186184(US9163013, 1)
Affinity DataIC50: 1.50E+3nMT: 2°CAssay Description:Compound 1 was also assayed to determine the IC50 values for three different kinases (PCTAIRE1, DYRK1a, and CDK2) in comparison to Gsk3beta. The assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186209BDBM186209(US9163013, 26)
Affinity DataIC50: 2.10E+3nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186184BDBM186184(US9163013, 1)
Affinity DataIC50: 2.90E+3nMT: 2°CAssay Description:Compound 1 was also assayed to determine the IC50 values for three different kinases (PCTAIRE1, DYRK1a, and CDK2) in comparison to Gsk3beta. The assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186214BDBM186214(US9163013, 31)
Affinity DataIC50: 7.20E+3nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent

TargetCyclin-dependent kinase 2(Human)
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandChemical structure of BindingDB Monomer ID 186184BDBM186184(US9163013, 1)
Affinity DataIC50: 3.60E+4nMT: 2°CAssay Description:Compound 1 was also assayed to determine the IC50 values for three different kinases (PCTAIRE1, DYRK1a, and CDK2) in comparison to Gsk3beta. The assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2016
Entry Details
US Patent