Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 7333
TargetSodium channel protein type 4 subunit alpha(Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190233BDBM190233(US9174999, Table 1, Compound 1)
Affinity DataIC50: 2.40nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha(Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190239BDBM190239(US9174999, Table 1, Compound 7)
Affinity DataIC50: 15nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha(Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190241BDBM190241(US9174999, 10)
Affinity DataIC50: 19nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha(Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190238BDBM190238(US9174999, Table 1, Compound 6)
Affinity DataIC50: 22.5nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha(Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190234BDBM190234(US9174999, 8)
Affinity DataIC50: 26nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha [I757A](Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190233BDBM190233(US9174999, Table 1, Compound 1)
Affinity DataIC50: 30nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha(Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 60830BDBM60830(US9174999, 13)
Affinity DataIC50: 46nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha(Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190237BDBM190237(US9174999, Table 1, Compound 5)
Affinity DataIC50: 55nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha(Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190240BDBM190240(US9174999, 9)
Affinity DataIC50: 83nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha(Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190243BDBM190243(US9174999, 12)
Affinity DataIC50: 87nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha [M1240A](Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190233BDBM190233(US9174999, Table 1, Compound 1)
Affinity DataIC50: 90nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha [I757A](Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190238BDBM190238(US9174999, Table 1, Compound 6)
Affinity DataIC50: 100nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha(Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190242BDBM190242(US9174999, 11)
Affinity DataIC50: 135nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha [I757A](Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190237BDBM190237(US9174999, Table 1, Compound 5)
Affinity DataIC50: 175nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha(Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190235BDBM190235(US9174999, Table 1, Compound 3 | US9174999, Table ...)
Affinity DataIC50: 230nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha [M1240A](Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190237BDBM190237(US9174999, Table 1, Compound 5)
Affinity DataIC50: 500nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha [M1240A](Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190238BDBM190238(US9174999, Table 1, Compound 6)
Affinity DataIC50: 500nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha [I757A](Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190235BDBM190235(US9174999, Table 1, Compound 3 | US9174999, Table ...)
Affinity DataIC50: 700nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha [M1240A](Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190235BDBM190235(US9174999, Table 1, Compound 3 | US9174999, Table ...)
Affinity DataIC50: 1.00E+3nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent

TargetSodium channel protein type 4 subunit alpha(Rat)
The Leland Stanford Junior University

US Patent
LigandChemical structure of BindingDB Monomer ID 190235BDBM190235(US9174999, Table 1, Compound 3 | US9174999, Table ...)
Affinity DataIC50: 6.00E+5nMAssay Description:In initial studies, we designed a set of molecules with branching at the nitrogen of the carbamate side chain as well as the carbon adjacent to the n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2016
Entry Details
US Patent