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Found 4 Enz. Inhib. hit(s) with all data for entry = 7361
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbvie

US Patent
LigandPNGBDBM50434335(CHEMBL2386729 | US9181275, 3)
Affinity DataKi:  0.0200nM ΔG°:  -61.1kJ/moleT: 2°CAssay Description:To determine the effectiveness of representative compounds of this invention as histamine-3 receptor ligands (H3 receptor ligands), the following tes...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbvie

US Patent
LigandPNGBDBM50434337(CHEMBL2386727 | US9181275, 1)
Affinity DataKi:  0.0320nM ΔG°:  -59.9kJ/moleT: 2°CAssay Description:To determine the effectiveness of representative compounds of this invention as histamine-3 receptor ligands (H3 receptor ligands), the following tes...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbvie

US Patent
LigandPNGBDBM50434336(CHEMBL2386728 | US9181275, 2)
Affinity DataKi:  0.0500nM ΔG°:  -58.8kJ/moleT: 2°CAssay Description:To determine the effectiveness of representative compounds of this invention as histamine-3 receptor ligands (H3 receptor ligands), the following tes...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbvie

US Patent
LigandPNGBDBM50434334(CHEMBL2386730 | US9181275, 4)
Affinity DataKi:  0.324nM ΔG°:  -54.2kJ/moleT: 2°CAssay Description:To determine the effectiveness of representative compounds of this invention as histamine-3 receptor ligands (H3 receptor ligands), the following tes...More data for this Ligand-Target Pair
In DepthDetails US Patent