Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 7403
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192902BDBM192902(US9193689, IQ-034)
Affinity DataIC50: 12nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192909BDBM192909(US9193689, IQ-222)
Affinity DataIC50: 16nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192904BDBM192904(US9193689, IQ-130)
Affinity DataIC50: 16nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192905BDBM192905(US9193689, REF-5)
Affinity DataIC50: 17nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192895BDBM192895(US9193689, IQ-025)
Affinity DataIC50: 17nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192903BDBM192903(US9193689, REF-4)
Affinity DataIC50: 18nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192899BDBM192899(US9193689, IQ-003)
Affinity DataIC50: 21nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192907BDBM192907(US9193689, REF-6)
Affinity DataIC50: 24nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192901BDBM192901(US9193689, REF-3)
Affinity DataIC50: 24nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192908BDBM192908(US9193689, IQ-220)
Affinity DataIC50: 26nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192897BDBM192897(US9193689, IQ-080)
Affinity DataIC50: 29nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192896BDBM192896(US9193689, REF-1)
Affinity DataIC50: 33nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192900BDBM192900(US9193689, IQ-002)
Affinity DataIC50: 39nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192912BDBM192912(US9193689, REF-8)
Affinity DataIC50: 39nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192910BDBM192910(US9193689, REF-7)
Affinity DataIC50: 42nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192898BDBM192898(US9193689, REF-2)
Affinity DataIC50: 48nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192906BDBM192906(US9193689, IQ-157)
Affinity DataIC50: 51nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192911BDBM192911(US9193689, IQ-223)
Affinity DataIC50: 76nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent