Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 7642
TargetCytochrome P450 2C9(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandPNGBDBM207974(US9266853, 5514403)
Affinity DataIC50: 7.70E+3nMT: 2°CAssay Description:Without Preincubation: To a 96 deep well plate was added 2.5 uL, of the test substance solution (x200 concentration), 442.5 uL of Incubation Mixture,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2017
Entry Details
US Patent

TargetCytochrome P450 3A4(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandPNGBDBM207975(US9266853, 5526064)
Affinity DataIC50: 1.18E+4nMT: 2°CAssay Description:With Preincubation: To a 96 deep well plate was added 2.5 uL of the test substance solution (x200 concentration), and 442.5 uL of Incubation Mixture,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2017
Entry Details
US Patent

TargetCytochrome P450 3A4(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandPNGBDBM207974(US9266853, 5514403)
Affinity DataIC50: 1.19E+4nMT: 2°CAssay Description:With Preincubation: To a 96 deep well plate was added 2.5 uL of the test substance solution (x200 concentration), and 442.5 uL of Incubation Mixture,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2017
Entry Details
US Patent

TargetCytochrome P450 2C9(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandPNGBDBM207975(US9266853, 5526064)
Affinity DataIC50: 1.25E+4nMT: 2°CAssay Description:Without Preincubation: To a 96 deep well plate was added 2.5 uL, of the test substance solution (x200 concentration), 442.5 uL of Incubation Mixture,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2017
Entry Details
US Patent

TargetCytochrome P450 3A4(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandPNGBDBM207975(US9266853, 5526064)
Affinity DataIC50: 1.62E+4nMT: 2°CAssay Description:Without Preincubation: To a 96 deep well plate was added 2.5 uL, of the test substance solution (x200 concentration), 442.5 uL of Incubation Mixture,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2017
Entry Details
US Patent

TargetCytochrome P450 2C9(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandPNGBDBM207974(US9266853, 5514403)
Affinity DataIC50: 1.96E+4nMT: 2°CAssay Description:With Preincubation: To a 96 deep well plate was added 2.5 uL of the test substance solution (x200 concentration), and 442.5 uL of Incubation Mixture,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2017
Entry Details
US Patent

TargetCytochrome P450 3A4(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandPNGBDBM207974(US9266853, 5514403)
Affinity DataIC50: 2.38E+4nMT: 2°CAssay Description:Without Preincubation: To a 96 deep well plate was added 2.5 uL, of the test substance solution (x200 concentration), 442.5 uL of Incubation Mixture,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2017
Entry Details
US Patent

TargetCytochrome P450 2C9(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandPNGBDBM207975(US9266853, 5526064)
Affinity DataIC50: 2.44E+4nMT: 2°CAssay Description:With Preincubation: To a 96 deep well plate was added 2.5 uL of the test substance solution (x200 concentration), and 442.5 uL of Incubation Mixture,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2017
Entry Details
US Patent