Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 8360
TargetHistone deacetylase 3(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 33.8nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242915(US9428447, DK-406)
Affinity DataIC50: 557nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 580nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242910(US9428447, DK-362)
Affinity DataIC50: 1.08E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242912(US9428447, DK-367)
Affinity DataIC50: 1.57E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242914(US9428447, DK-405)
Affinity DataIC50: 1.97E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242906(US9428447, DK-319)
Affinity DataIC50: 2.65E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242913(US9428447, DK-381)
Affinity DataIC50: 3.13E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242909(US9428447, DK-361)
Affinity DataIC50: 3.40E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242908(US9428447, DK-347)
Affinity DataIC50: 3.94E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242916(US9428447, JF-B06)
Affinity DataIC50: 4.70E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242907(US9428447, DK-320)
Affinity DataIC50: 5.03E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242911(US9428447, DK-366)
Affinity DataIC50: 7.40E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 3(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242901(US9428447, JFD-15)
Affinity DataIC50: 9.83E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 3(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242899(US9428447, JF-B53)
Affinity DataIC50: 1.70E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 3(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242898(US9428447, JF-C71)
Affinity DataIC50: 2.20E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242903(US9428447, DK-178)
Affinity DataIC50: 2.49E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242898(US9428447, JF-C71)
Affinity DataIC50: 2.61E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242905(US9428447, DK-305)
Affinity DataIC50: 2.92E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 3(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242900(US9428447, JF-B54)
Affinity DataIC50: 2.99E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 3(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242904(US9428447, DK-201)
Affinity DataIC50: 3.05E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242900(US9428447, JF-B54)
Affinity DataIC50: 3.15E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242899(US9428447, JF-B53)
Affinity DataIC50: 3.33E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242902(US9428447, JFD-50)
Affinity DataIC50: 3.61E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 3(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242917(US9428447, JF-B21)
Affinity DataIC50: 3.61E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242917(US9428447, JF-B21)
Affinity DataIC50: 3.79E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 3(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242902(US9428447, JFD-50)
Affinity DataIC50: 4.51E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 6(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242901(US9428447, JFD-15)
Affinity DataIC50: 4.71E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetHistone deacetylase 3(Human)
The Royal Institution For The Advancement of Learning/Mcgill University

US Patent
LigandPNGBDBM242903(US9428447, DK-178)
Affinity DataIC50: 4.73E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent