Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 8558
TargetCytochrome P450 3A4(Human)
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM258443(US9512130, 1 | US11208696, Example 6)
Affinity DataIC50: 5.00E+3nMpH: 7.4 T: 2°CAssay Description:The potential of the test compound to act as a competitive inhibitor of CYP3A4 was evaluated in in vitro assays, using human liver microsomes and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2017
Entry Details
US Patent

TargetCytochrome P450 3A4(Human)
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM258445(US9512130, 3 | US11208696, Example 5)
Affinity DataIC50: 1.00E+4nMpH: 7.4 T: 2°CAssay Description:The potential of the test compound to act as a competitive inhibitor of CYP3A4 was evaluated in in vitro assays, using human liver microsomes and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2017
Entry Details
US Patent

TargetCytochrome P450 3A4(Human)
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM258446(US9512130, Ref.)
Affinity DataIC50: 1.00E+4nMpH: 7.4 T: 2°CAssay Description:The potential of the test compound to act as a competitive inhibitor of CYP3A4 was evaluated in in vitro assays, using human liver microsomes and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2017
Entry Details
US Patent

TargetCytochrome P450 3A4(Human)
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM258444(US9512130, 2)
Affinity DataIC50: 1.00E+4nMpH: 7.4 T: 2°CAssay Description:The potential of the test compound to act as a competitive inhibitor of CYP3A4 was evaluated in in vitro assays, using human liver microsomes and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2017
Entry Details
US Patent