Compile Data Set for Download or QSAR
Report error Found 191 Enz. Inhib. hit(s) with all data for entry = 152
LigandPNGBDBM195729(US9670212, 119 3-iodo-1-{[5-methyl-3-(2-methylphen...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195724(US9670212, 117 3-iodo-1-{1-[3-(2-methylphenyl)quin...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195361(US9670212, 48 3-amino-N-[(5-chloro-3-{2-[(dimethyl...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195082(US9670212, 3 3-[(6-amino-9H-purin-9-yl)methyl]-N,8...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195452(US9670212, 67 3-amino-N-{[8-methyl-2-(methyl{2-[me...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM50004540(CHEMBL2216869 | US9670212, 2 3-[(6-amino-9H-purin-...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195740(US9670212, 128 3-amino-N-[(2-{[2-(dimethylamino)et...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195468(US9670212, 73 3-amino-N-({8-methyl-2-[methyl(2-{me...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195759(US9670212, 136 3-amino-N-({2-[{3-[(N,N-dimethylgly...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195755(US9670212, 134 3-iodo-1-{[8-methyl-2-(2-methylphen...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195083(US9670212, 4 3-[(6-amino-9H-purin-9-yl)methyl]-N,8...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195625(US9670212, 83 3-amino-N-{[8-methyl-2-(methyl{2-[me...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195785(US9670212, 146 N-{[8-methyl-2-(4-methyl-1,4-diazep...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195784(US9670212, 145 3-iodo-1-{[3-(2-methylphenyl)quinol...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195783(US9670212, 144 N-{[2-(4-ethylpiperazin-1-yl)-8-met...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195767(US9670212, 143 N-{[2-(4-acetylpiperazin-1-yl)-8-me...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195165(US9670212, 12 N-{[8-methyl-2-(octahydro-2H-pyrido[...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195793(US9670212, 154 N-{[2-(2-chlorophenyl)-8-methylquin...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195214(US9670212, 25 N,8-dimethyl-N-[2-(methyloxy)ethyl]-...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195636(US9670212, 89 3-amino-N-({2-[(2-{[2-(dimethylamino...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195791(US9670212, 152 N-{1-[2-(2-chlorophenyl)-8-methylqu...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195632(US9670212, 86 3-amino-N-({8-methyl-2-[methyl(2-{me...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195631(US9670212, 85 3-amino-N-({2-[{2-[(1H-imidazol-1-yl...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195788(US9670212, 149 N-{3-[(6-amino-9H-purin-9-yl)methyl...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195302(US9670212, 35 N-methyl-N-[2-(methyl{8-methyl-3-[(9...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195289(US9670212, 34 N-{2-[{3-[(6-amino-9H-purin-9-yl)met...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195271(US9670212, 33 N,8-dimethyl-N-[(1-methylpiperidin-4...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195256(US9670212, 32 N,8-dimethyl-N-[(1-methylpiperidin-3...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195254(US9670212, 31 3-amino-N-[(8-methyl-2-{methyl[(1-me...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195234(US9670212, 30 3-amino-N-[(8-methyl-2-{methyl[(1-me...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195231(US9670212, 28 N-{2-[{3-[(6-amino-9H-purin-9-yl)met...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195341(US9670212, 43 3-amino-N-({2-[(2-{[(3,5-dimethyl-1H...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195333(US9670212, 42 3-amino-N-{[8-methyl-2-(methyl{2-[me...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195323(US9670212, 39 3-amino-N-[(8-methyl-2-{methyl[(1-me...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195315(US9670212, 38 N,8-dimethyl-N-[(1-methylpiperidin-2...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195314(US9670212, 37 N-[(8-methyl-2-piperazin-1-ylquinoli...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195313(US9670212, 36 N,N'-dimethyl-N-{8-methyl-3-[(9H-pur...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195664(US9670212, 100 3-amino-N-{[8-methyl-2-(methyl{2-[m...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195364(US9670212, 49 3-amino-N-{[8-methyl-2-(methyl{2-[me...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195361(US9670212, 48 3-amino-N-[(5-chloro-3-{2-[(dimethyl...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195823(US9670212, 175 3-amino-N-{[5-methyl-3-(2-methylphe...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195852(US9670212, 187 9-{[2-(2-chlorophenyl)-8-methylquin...)
Affinity DataIC50: 150nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195444(US9670212, 59 3-amino-N-({3-[2-(piperidin-1-ylmeth...)
Affinity DataIC50: 150nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195731(US9670212, 121 3-amino-N-({2-[(2-hydroxyethyl)(met...)
Affinity DataIC50: 150nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195847(US9670212, 182 9-({8-methyl-2-[2-(trifluoromethyl)...)
Affinity DataIC50: 150nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195846(US9670212, 181 9-{[2-(2,5-dimethylphenyl)-8-methyl...)
Affinity DataIC50: 150nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195723(US9670212, 116 3-amino-N-{[8-methyl-2-(methyl{2-[m...)
Affinity DataIC50: 150nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195080(US9670212, 1 N,8-dimethyl-N-[(1-methylpiperidin-4-...)
Affinity DataIC50: 150nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195448(US9670212, 63 3-amino-N-[(8-methyl-2-{4-[(1-methyl...)
Affinity DataIC50: 150nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

LigandPNGBDBM195854(US9670212, 189 9-{[8-methyl-2-(2-methylphenyl)quin...)
Affinity DataIC50: 150nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

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