Compile Data Set for Download or QSAR
Report error Found 91 Enz. Inhib. hit(s) with all data for entry = 260
TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261601(US9708270, 107)
Affinity DataEC50:  202nMAssay Description:IP1 assay results were obtained adapting the GPR120 assay described in C. Bergsdorf, et al., Assay Drug Dev. Technol., 2008, 6(1), 39-53.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261600(US9708270, 106)
Affinity DataEC50:  220nMAssay Description:IP1 assay results were obtained adapting the GPR120 assay described in C. Bergsdorf, et al., Assay Drug Dev. Technol., 2008, 6(1), 39-53.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261552(US9708270, 47)
Affinity DataEC50:  330nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261553(US9708270, 48)
Affinity DataEC50:  377nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM50208148(US9708270, 7 | CHEMBL3891920)
Affinity DataEC50:  410nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM50208154(US9708270, 35 | CHEMBL3973034)
Affinity DataEC50:  431nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261554(US9708270, 49)
Affinity DataEC50:  449nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM50208152(US9708270, 50 | CHEMBL3967504)
Affinity DataEC50:  472nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261523(US9708270, 18)
Affinity DataEC50:  530nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261556(US9708270, 51)
Affinity DataEC50:  617nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261557(US9708270, 52)
Affinity DataEC50:  641nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM50208150(US9708270, 16 | CHEMBL3947837)
Affinity DataEC50:  652nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261558(US9708270, 53)
Affinity DataEC50:  667nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261539(US9708270, 34)
Affinity DataEC50:  671nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261559(US9708270, 54)
Affinity DataEC50:  681nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261547(US9708270, 42)
Affinity DataEC50:  749nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261541(US9708270, 36)
Affinity DataEC50:  832nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261560(US9708270, 55)
Affinity DataEC50:  869nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM50208157(US9708270, 30 | CHEMBL3893026)
Affinity DataEC50:  878nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261524(US9708270, 19)
Affinity DataEC50:  948nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM50208093(US9708270, 25 | CHEMBL3953289)
Affinity DataEC50:  1.15E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261550(US9708270, 45)
Affinity DataEC50:  1.17E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261592(US9708270, 96)
Affinity DataEC50:  1.21E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261561(US9708270, 56)
Affinity DataEC50:  1.22E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261536(US9708270, 31)
Affinity DataEC50:  1.22E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261551(US9708270, 46)
Affinity DataEC50:  1.29E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM50208151(US9708270, 97 | CHEMBL3986483)
Affinity DataEC50:  1.29E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261562(US9708270, 57)
Affinity DataEC50:  1.33E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261587(US9708270, 84)
Affinity DataEC50:  1.35E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261563(US9708270, 58)
Affinity DataEC50:  1.44E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261564(US9708270, 59)
Affinity DataEC50:  1.49E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261594(US9708270, 98)
Affinity DataEC50:  1.53E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261565(US9708270, 60)
Affinity DataEC50:  1.55E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261595(US9708270, 99)
Affinity DataEC50:  1.65E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261525(US9708270, 20)
Affinity DataEC50:  1.66E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM50208084(US9708270, 8 | CHEMBL3977361)
Affinity DataEC50:  1.67E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261546(US9708270, 41)
Affinity DataEC50:  1.69E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261515(US9708270, 10)
Affinity DataEC50:  1.70E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261534(US9708270, 29)
Affinity DataEC50:  1.79E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM50208094(US9708270, 85 | CHEMBL3897637)
Affinity DataEC50:  1.79E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261544(US9708270, 39)
Affinity DataEC50:  1.80E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261591(US9708270, 95)
Affinity DataEC50:  1.90E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261566(US9708270, 61)
Affinity DataEC50:  1.96E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261589(US9708270, 86)
Affinity DataEC50:  2.02E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261518(US9708270, 13)
Affinity DataEC50:  2.14E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM50208146(US9708270, 38 | CHEMBL3901994)
Affinity DataEC50:  2.15E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261567(US9708270, 62)
Affinity DataEC50:  2.15E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261537(US9708270, 32)
Affinity DataEC50:  2.15E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261542(US9708270, 37)
Affinity DataEC50:  2.17E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM261514(US9708270, 9)
Affinity DataEC50:  2.18E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

Displayed 1 to 50 (of 91 total ) | Next | Last >>
Jump to: