Compile Data Set for Download or QSAR
Report error Found 257 Enz. Inhib. hit(s) with all data for entry = 390
LigandChemical structure of BindingDB Monomer ID 264615BDBM264615(US9718760, C182)
Affinity DataIC50: 33nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264650BDBM264650(US9718760, C204)
Affinity DataIC50: 35nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264630BDBM264630(US9718760, C198)
Affinity DataIC50: 51nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264611BDBM264611(US9718760, C188)
Affinity DataIC50: 120nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264602BDBM264602(US9718760, C197)
Affinity DataIC50: 173nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264616BDBM264616(US9718760, C183)
Affinity DataIC50: 180nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264613BDBM264613(US9718760, C157)
Affinity DataIC50: 250nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264609BDBM264609(US9718760, C163)
Affinity DataIC50: 288nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264610BDBM264610(US9718760, C165)
Affinity DataIC50: 350nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264645BDBM264645(US9718760, C185)
Affinity DataIC50: 420nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264646BDBM264646(US9718760, C196)
Affinity DataIC50: 450nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetPlasminogen activator inhibitor 1/Tissue-type plasminogen activator(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 264610BDBM264610(US9718760, C165)
Affinity DataIC50: 510nMT: 2°CAssay Description:PAI-1 inhibitor compounds were dissolved in DMSO to a final concentration of (10-50 mM), depending upon solubility. Compounds were then diluted in ph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264644BDBM264644(US9718760, C184)
Affinity DataIC50: 590nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetPlasminogen activator inhibitor 1/Tissue-type plasminogen activator(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 264609BDBM264609(US9718760, C163)
Affinity DataIC50: 611nMT: 2°CAssay Description:PAI-1 inhibitor compounds were dissolved in DMSO to a final concentration of (10-50 mM), depending upon solubility. Compounds were then diluted in ph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264643BDBM264643(US9718760, C176)
Affinity DataIC50: 620nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264607BDBM264607(US9718760, C153)
Affinity DataIC50: 700nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264628BDBM264628(US9718760, C187)
Affinity DataIC50: 910nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264612BDBM264612(US9718760, C195)
Affinity DataIC50: 920nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetPlasminogen activator inhibitor 1/Tissue-type plasminogen activator(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 264613BDBM264613(US9718760, C157)
Affinity DataIC50: 980nMT: 2°CAssay Description:PAI-1 inhibitor compounds were dissolved in DMSO to a final concentration of (10-50 mM), depending upon solubility. Compounds were then diluted in ph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetPlasminogen activator inhibitor 1/Tissue-type plasminogen activator(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 264607BDBM264607(US9718760, C153)
Affinity DataIC50: 1.02E+3nMT: 2°CAssay Description:PAI-1 inhibitor compounds were dissolved in DMSO to a final concentration of (10-50 mM), depending upon solubility. Compounds were then diluted in ph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264601BDBM264601(US9718760, C191)
Affinity DataIC50: 1.28E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264623BDBM264623(US9718760, C180)
Affinity DataIC50: 1.34E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetPlasminogen activator inhibitor 1/Tissue-type plasminogen activator(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 264614BDBM264614(US9718760, C158)
Affinity DataIC50: 1.44E+3nMT: 2°CAssay Description:PAI-1 inhibitor compounds were dissolved in DMSO to a final concentration of (10-50 mM), depending upon solubility. Compounds were then diluted in ph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264597BDBM264597(US9718760, C152)
Affinity DataIC50: 1.57E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264618BDBM264618(US9718760, C171)
Affinity DataIC50: 1.67E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetPlasminogen activator inhibitor 1/Tissue-type plasminogen activator(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 264597BDBM264597(US9718760, C152)
Affinity DataIC50: 1.71E+3nMT: 2°CAssay Description:PAI-1 inhibitor compounds were dissolved in DMSO to a final concentration of (10-50 mM), depending upon solubility. Compounds were then diluted in ph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264635BDBM264635(US9718760, C271)
Affinity DataIC50: 1.82E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264642BDBM264642(US9718760, C168)
Affinity DataIC50: 1.98E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264619BDBM264619(US9718760, C172)
Affinity DataIC50: 1.98E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetPlasminogen activator inhibitor 1/Tissue-type plasminogen activator(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 264648BDBM264648(US9718760, C161)
Affinity DataIC50: 2.21E+3nMT: 2°CAssay Description:PAI-1 inhibitor compounds were dissolved in DMSO to a final concentration of (10-50 mM), depending upon solubility. Compounds were then diluted in ph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264600BDBM264600(US9718760, C189)
Affinity DataIC50: 2.29E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264622BDBM264622(US9718760, C179)
Affinity DataIC50: 2.40E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264614BDBM264614(US9718760, C158)
Affinity DataIC50: 2.60E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264648BDBM264648(US9718760, C161)
Affinity DataIC50: 3.70E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264608BDBM264608(US9718760, C162)
Affinity DataIC50: 3.90E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264603BDBM264603(US9718760, C224)
Affinity DataIC50: 4.34E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264660BDBM264660(US9718760, C206)
Affinity DataIC50: 4.96E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264626BDBM264626(US9718760, C205)
Affinity DataIC50: 5.05E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264621BDBM264621(US9718760, C177)
Affinity DataIC50: 5.11E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264658BDBM264658(US9718760, C199)
Affinity DataIC50: 5.36E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264617BDBM264617(US9718760, C170)
Affinity DataIC50: 5.49E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264620BDBM264620(US9718760, C175)
Affinity DataIC50: 6.74E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264624BDBM264624(US9718760, C186)
Affinity DataIC50: 6.98E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetPlasminogen activator inhibitor 1/Tissue-type plasminogen activator(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 264608BDBM264608(US9718760, C162)
Affinity DataIC50: 7.59E+3nMT: 2°CAssay Description:PAI-1 inhibitor compounds were dissolved in DMSO to a final concentration of (10-50 mM), depending upon solubility. Compounds were then diluted in ph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264629BDBM264629(US9718760, C190)
Affinity DataIC50: 9.70E+3nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264640BDBM264640(US9718760, C303)
Affinity DataIC50: 1.26E+4nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264631BDBM264631(US9718760, C232)
Affinity DataIC50: 1.33E+4nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264664BDBM264664(US9718760, C228)
Affinity DataIC50: 1.48E+4nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264636BDBM264636(US9718760, C272)
Affinity DataIC50: 1.64E+4nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 264661BDBM264661(US9718760, C207)
Affinity DataIC50: 1.68E+4nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

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