Compile Data Set for Download or QSAR
Report error Found 224 Enz. Inhib. hit(s) with all data for entry = 2278
TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360269BDBM360269((S)-(1-methyl- | US9828339, Example 174)
Affinity DataKi:  0.610nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360258BDBM360258((S)-(1-methyl- | US9828339, Example 165)
Affinity DataKi:  0.630nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360292BDBM360292((S)-(1-methylpyrrolidin-2-yl)-methyl [1,1'-bipheny...)
Affinity DataKi:  0.780nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360189BDBM360189((S)-(1-ethylpyrrolidin-2-yl)methyl [1,1'-biphenyl]...)
Affinity DataKi:  0.800nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360294BDBM360294((S)-(1-methyl- | US9828339, Example 199)
Affinity DataKi:  0.800nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360045BDBM360045(3',5-Difluoro- | US9828339, Example 17)
Affinity DataKi:  1nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360290BDBM360290((R)-(1-methyl- | US9828339, Example 195)
Affinity DataKi:  1.08nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360227BDBM360227((R)-(1-methyl- | US9828339, Example 143)
Affinity DataKi:  1.12nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360036BDBM360036(3',5'-Dichloro-[1,1'- | US9828339, Example 8)
Affinity DataKi:  1.33nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360101BDBM360101(2-(1-Methyl- | US9828339, Example 53)
Affinity DataKi:  1.34nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360091BDBM360091(2-(1-Methyl- | US9828339, Example 43)
Affinity DataKi:  1.48nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360235BDBM360235((S)-(1-methyl- | US9828339, Example 149)
Affinity DataKi:  1.57nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360220BDBM360220((R)-(1-methylpyrrolidin-3-yl)-methyl (3'-chloro-4'...)
Affinity DataKi:  1.59nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360201BDBM360201((R)-(1-methyl- | US9828339, Example 117)
Affinity DataKi:  1.60nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360205BDBM360205((S)-(1-methyl- | US9828339, Example 121)
Affinity DataKi:  1.75nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360293BDBM360293((S)-(1-methyl- | US9828339, Example 198)
Affinity DataKi:  1.87nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360196BDBM360196((R)-(1-methylpyrrolidin-3-yl)-methyl (3'-fluoro-[1...)
Affinity DataKi:  1.92nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360156BDBM360156((S)-(1-methylpyrrolidin- | US9828339, Example 90)
Affinity DataKi:  1.97nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360295BDBM360295((S)-(1-methyl- | US9828339, Example 200)
Affinity DataKi:  2.03nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360214BDBM360214((R)-(1-methylpyrrolidin-3-yl)-methyl (3',4'-dichlo...)
Affinity DataKi:  2.10nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360285BDBM360285((S)-(1-methyl- | US9828339, Example 190)
Affinity DataKi:  2.17nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360297BDBM360297((S)-(1-methyl- | US9828339, Example 202)
Affinity DataKi:  2.18nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360055BDBM360055(5-Fluoro-3'- | US9828339, Example 21)
Affinity DataKi:  2.25nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360043BDBM360043(3'-Ethoxy-[1,1'- | US9828339, Example 15)
Affinity DataKi:  2.27nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360298BDBM360298((S)-(1-methyl- | US9828339, Example 203)
Affinity DataKi:  2.36nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360202BDBM360202((S)-(1-methyl- | US9828339, Example 118)
Affinity DataKi:  2.42nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360155BDBM360155((R)-(1-methylpyrrolidin-3-yl)methyl [1,1'-biphenyl...)
Affinity DataKi:  2.43nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360180BDBM360180((R)-(1-methylpyrrolidin-3-yl)methyl(3'-methyl-[1,1...)
Affinity DataKi:  2.43nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360087BDBM360087(2-(1-Methyl- | US9828339, Example 41)
Affinity DataKi:  2.45nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360034BDBM360034(4'-Chloro-[1,1'- | US9828339, Example 6)
Affinity DataKi:  2.47nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360209BDBM360209((S)-(1-methyl- | US9828339, Example 125)
Affinity DataKi:  2.67nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360296BDBM360296((S)-(1-methyl- | US9828339, Example 201)
Affinity DataKi:  2.70nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360032BDBM360032(3'-Fluoro-[1,1'- | US9828339, Example 4)
Affinity DataKi:  2.93nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360276BDBM360276((S)-(1-methyl- | US9828339, Example 181)
Affinity DataKi:  3.29nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360212BDBM360212((S)-(1-methyl- | US9828339, Example 128)
Affinity DataKi:  3.41nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360299BDBM360299((S)-(1-methyl- | US9828339, Example 204)
Affinity DataKi:  3.53nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360195BDBM360195((S)-(1-isopropylpyrrolidin-2-yl)-methyl [1,1'-biph...)
Affinity DataKi:  3.77nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360056BDBM360056(4-Fluoro-[1,1'- | US9828339, Example 22)
Affinity DataKi:  3.79nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360182BDBM360182((S)-(1-methylpyrrolidin-3-yl)-methyl(3'-methyl-[1,...)
Affinity DataKi:  3.79nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360191BDBM360191((S)-(1-methylpyrrolidin-3-yl)-methyl(3',5-difluoro...)
Affinity DataKi:  3.95nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360173BDBM360173((S)-(1-methylpyrrolidin- | US9828339, Example 93)
Affinity DataKi:  4.12nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360047BDBM360047(3',5,5'- | US9828339, Example 19)
Affinity DataKi:  4.17nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360198BDBM360198((R)-(1-methyl- | US9828339, Example 114)
Affinity DataKi:  4.23nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360250BDBM360250((S)-(1-methyl- | US9828339, Example 160)
Affinity DataKi:  4.29nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360028BDBM360028(4'-Fluoro-[1,1'- | US9828339, Example 1)
Affinity DataKi:  4.42nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360157BDBM360157((R)-(1-methylpyrrolidin- | US9828339, Example 91)
Affinity DataKi:  4.5nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360287BDBM360287((R)-(1-methyl- | US9828339, Example 192)
Affinity DataKi:  4.60nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360305BDBM360305((S)-(1-methyl- | US9828339, Example 210)
Affinity DataKi:  4.60nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360144BDBM360144((R)-pyrrolidin-3-ylmethyl [1,1'-biphenyl]-2-ylcarb...)
Affinity DataKi:  4.62nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 360216BDBM360216((R)-(1-methyl- | US9828339, Example 132)
Affinity DataKi:  4.64nMAssay Description:Cell membrane proteins (Perkin Elmer) wherein human muscarinic M3 receptor was overexpressed, [3H]-methyl scopolamine and test compounds in various c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details
US Patent

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