Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 2400
TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364218BDBM364218(US9856263, 1 | US9856263, 3 | US9856263, 2)
Affinity DataKi:  4.5nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364218BDBM364218(US9856263, 1 | US9856263, 3 | US9856263, 2)
Affinity DataKi:  5.5nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364363BDBM364363(US9856263, 15)
Affinity DataKi:  7.30nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364317BDBM364317(US9856263, 37)
Affinity DataKi:  12.7nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364293BDBM364293(US9856263, 13 | (+)-1-[4-(3,5-Dimethylpyridazin-4-...)
Affinity DataKi:  13.1nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364362BDBM364362(US9856263, 14)
Affinity DataKi:  18.8nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364218BDBM364218(US9856263, 1 | US9856263, 3 | US9856263, 2)
Affinity DataKi:  20.5nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364284BDBM364284(US9856263, 4 | 1-[4-(4, 6-Dimethylpyrimidin-5-yl)-...)
Affinity DataKi:  22.1nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364307BDBM364307(US9856263, 27)
Affinity DataKi:  28.1nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364319BDBM364319(US9856263, 39)
Affinity DataKi:  31.2nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364315BDBM364315(US9856263, 35)
Affinity DataKi:  31.5nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364321BDBM364321(US9856263, 41)
Affinity DataKi:  34.7nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364289BDBM364289(US9856263, 9 | 4-[4-(3,5-Dimethylpyridazin-4-yl)-3...)
Affinity DataKi:  35.8nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364316BDBM364316(US9856263, 36)
Affinity DataKi:  48.7nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364314BDBM364314(US9856263, 34)
Affinity DataKi:  49.4nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364285BDBM364285(US9856263, 5 | 4-[4-(4,6-Dimethylpyrimidin-5-yl)-3...)
Affinity DataKi:  56.4nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364305BDBM364305(US9856263, 25)
Affinity DataKi:  56.4nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364296BDBM364296(US9856263, 16)
Affinity DataKi:  58.2nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364310BDBM364310(US9856263, 30)
Affinity DataKi:  59nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364300BDBM364300(US9856263, 20)
Affinity DataKi:  59.3nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364286BDBM364286(US9856263, 6 | 4-[4-(4, 6-Dimethylpyrimidin-5-yl)-...)
Affinity DataKi:  61.3nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364290BDBM364290(US9856263, 10 | 2-(4,6-Dimethylpyrimidin-5-yl)-5-(...)
Affinity DataKi:  63.9nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364304BDBM364304(US9856263, 24)
Affinity DataKi:  83.9nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364309BDBM364309(US9856263, 29)
Affinity DataKi:  85.7nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364306BDBM364306(US9856263, 26)
Affinity DataKi:  86.1nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364292BDBM364292(US9856263, 12 | (-)-1-[4-(3,5-Dimethylpyridazin-4-...)
Affinity DataKi:  96.3nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364301BDBM364301(US9856263, 21)
Affinity DataKi:  102nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364302BDBM364302(US9856263, 22)
Affinity DataKi:  105nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364288BDBM364288(US9856263, 8 | 6-Methyl-5-[2-methyl-4-(pyrazolo[1,...)
Affinity DataKi:  107nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364312BDBM364312(US9856263, 32)
Affinity DataKi:  116nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364318BDBM364318(US9856263, 38)
Affinity DataKi:  141nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364311BDBM364311(US9856263, 31)
Affinity DataKi:  179nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364297BDBM364297(US9856263, 17)
Affinity DataKi:  183nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364308BDBM364308(US9856263, 28)
Affinity DataKi:  198nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364313BDBM364313(US9856263, 33)
Affinity DataKi:  252nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364287BDBM364287(US9856263, 7 | 4-[4-(4, 6-Dimethylpyrimidin-5-yl)p...)
Affinity DataKi:  514nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364299BDBM364299(US9856263, 19)
Affinity DataKi:  672nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364303BDBM364303(US9856263, 23)
Affinity DataKi:  894nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364298BDBM364298(US9856263, 18)
Affinity DataKi:  1.15E+3nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364361BDBM364361(US9856263, 11)
Affinity DataKi:  1.82E+3nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 364320BDBM364320(US9856263, 40)
Affinity DataKi: >6.40E+3nMAssay Description:Frozen cells were quickly thawed, re-suspended in 50 mL warm media and allowed to sit for 5 min prior to centrifugation (1000 rpm) at room temperatur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent