Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 2624
TargetVascular endothelial growth factor receptor 2(Human)
Peking University Founder Group

US Patent
LigandChemical structure of BindingDB Monomer ID 373143BDBM373143(FD-2013015 | US9902709, Compound Example 1)
Affinity DataIC50: 28.6nMAssay Description:Kinase Enzymatic step assay Control (10 μL) Sample Negative Positive Compound 4 μL 4 μL 2.5% 4 μL 2.5% DMSO/kinase DMSO/kinase bu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
Peking University Founder Group

US Patent
LigandChemical structure of BindingDB Monomer ID 373144BDBM373144(FD-2013018 | US9902709, Compound Example 2)
Affinity DataIC50: 55.5nMAssay Description:Kinase Enzymatic step assay Control (10 μL) Sample Negative Positive Compound 4 μL 4 μL 2.5% 4 μL 2.5% DMSO/kinase DMSO/kinase bu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
Peking University Founder Group

US Patent
LigandChemical structure of BindingDB Monomer ID 373202BDBM373202(FD-2013025 | US9902709, Compound Example 4)
Affinity DataIC50: 68.5nMAssay Description:Kinase Enzymatic step assay Control (10 μL) Sample Negative Positive Compound 4 μL 4 μL 2.5% 4 μL 2.5% DMSO/kinase DMSO/kinase bu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
Peking University Founder Group

US Patent
LigandChemical structure of BindingDB Monomer ID 16673BDBM16673(BAY439006 | CHEMBL1336 | BAY 43-9006 | 4-[4-({[4-c...)
Affinity DataIC50: 89.6nMAssay Description:Kinase Enzymatic step assay Control (10 μL) Sample Negative Positive Compound 4 μL 4 μL 2.5% 4 μL 2.5% DMSO/kinase DMSO/kinase bu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetVascular endothelial growth factor receptor 2(Human)
Peking University Founder Group

US Patent
LigandChemical structure of BindingDB Monomer ID 373275BDBM373275(FD-1210005 | US9902709, Comparative example 2)
Affinity DataIC50: 188nMAssay Description:Kinase Enzymatic step assay Control (10 μL) Sample Negative Positive Compound 4 μL 4 μL 2.5% 4 μL 2.5% DMSO/kinase DMSO/kinase bu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
Peking University Founder Group

US Patent
LigandChemical structure of BindingDB Monomer ID 373262BDBM373262(FD-2013031 | US9902709, Compound Example 6)
Affinity DataIC50: 215nMAssay Description:Kinase Enzymatic step assay Control (10 μL) Sample Negative Positive Compound 4 μL 4 μL 2.5% 4 μL 2.5% DMSO/kinase DMSO/kinase bu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
Peking University Founder Group

US Patent
LigandChemical structure of BindingDB Monomer ID 373150BDBM373150(FD-2013024 | US9902709, Compound Example 3)
Affinity DataIC50: 222nMAssay Description:Kinase Enzymatic step assay Control (10 μL) Sample Negative Positive Compound 4 μL 4 μL 2.5% 4 μL 2.5% DMSO/kinase DMSO/kinase bu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
Peking University Founder Group

US Patent
LigandChemical structure of BindingDB Monomer ID 373261BDBM373261(FD-2013027 | US9902709, Compound Example 5)
Affinity DataIC50: 317nMAssay Description:Kinase Enzymatic step assay Control (10 μL) Sample Negative Positive Compound 4 μL 4 μL 2.5% 4 μL 2.5% DMSO/kinase DMSO/kinase bu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
Peking University Founder Group

US Patent
LigandChemical structure of BindingDB Monomer ID 373273BDBM373273(FD-2013037 | US9902709, Compound Example 8)
Affinity DataIC50: 417nMAssay Description:Kinase Enzymatic step assay Control (10 μL) Sample Negative Positive Compound 4 μL 4 μL 2.5% 4 μL 2.5% DMSO/kinase DMSO/kinase bu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
Peking University Founder Group

US Patent
LigandChemical structure of BindingDB Monomer ID 373516BDBM373516(FD-2013016 | US9902709, Comparative example 3)
Affinity DataIC50: 437nMAssay Description:Kinase Enzymatic step assay Control (10 μL) Sample Negative Positive Compound 4 μL 4 μL 2.5% 4 μL 2.5% DMSO/kinase DMSO/kinase bu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
Peking University Founder Group

US Patent
LigandChemical structure of BindingDB Monomer ID 373272BDBM373272(FD-2013033 | US9902709, Compound Example 7)
Affinity DataIC50: 656nMAssay Description:Kinase Enzymatic step assay Control (10 μL) Sample Negative Positive Compound 4 μL 4 μL 2.5% 4 μL 2.5% DMSO/kinase DMSO/kinase bu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
Peking University Founder Group

US Patent
LigandChemical structure of BindingDB Monomer ID 373518BDBM373518(FD-2013017 | US9902709, Comparative example 5)
Affinity DataIC50: 2.39E+3nMAssay Description:Kinase Enzymatic step assay Control (10 μL) Sample Negative Positive Compound 4 μL 4 μL 2.5% 4 μL 2.5% DMSO/kinase DMSO/kinase bu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
Peking University Founder Group

US Patent
LigandChemical structure of BindingDB Monomer ID 373517BDBM373517(FD-2013019 | US9902709, Comparative example 4)
Affinity DataIC50: 2.05E+4nMAssay Description:Kinase Enzymatic step assay Control (10 μL) Sample Negative Positive Compound 4 μL 4 μL 2.5% 4 μL 2.5% DMSO/kinase DMSO/kinase bu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent