Compile Data Set for Download or QSAR
Report error Found 488 Enz. Inhib. hit(s) with all data for entry = 3049
LigandChemical structure of BindingDB Monomer ID 293423BDBM293423(US10106527, Compound 461 | US10106527, Compound 9 ...)
Affinity DataEC50:  0.400nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293564BDBM293564(US10106527, Compound 275 | US9951048, Compound 275...)
Affinity DataEC50:  0.600nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293619BDBM293619(US10106527, Compound 391 | US9951048, Compound 391...)
Affinity DataEC50:  0.700nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293479BDBM293479(US10106527, Compound 93 | US9951048, Compound 93 |...)
Affinity DataEC50:  0.700nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293566BDBM293566(US10106527, Compound 277 | US9951048, Compound 277...)
Affinity DataEC50:  0.800nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293415BDBM293415(US10106527, Compound 145 | US10106527, Compound 1 ...)
Affinity DataEC50:  0.800nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293569BDBM293569(US10106527, Compound 286 | US9951048, Compound 286...)
Affinity DataEC50:  0.800nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293616BDBM293616(US10106527, Compound 388 | US9951048, Compound 388...)
Affinity DataEC50:  0.800nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293422BDBM293422(US10106527, Compound 8 | US9951048, Compound 8 | U...)
Affinity DataEC50:  0.900nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293613BDBM293613(US10106527, Compound 385 | US9951048, Compound 385...)
Affinity DataEC50:  0.900nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293428BDBM293428(US10106527, Compound 14 | US9951048, Compound 14 |...)
Affinity DataEC50:  0.900nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293444BDBM293444(US10106527, Compound 37 | US9951048, Compound 37 |...)
Affinity DataEC50:  0.900nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293417BDBM293417(US10106527, Compound 3 | US9951048, Compound 3 | U...)
Affinity DataEC50:  0.900nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293577BDBM293577(US10106527, Compound 301 | US9951048, Compound 301...)
Affinity DataEC50:  0.900nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293597BDBM293597(US10106527, Compound 338 | US9951048, Compound 338...)
Affinity DataEC50:  1nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Samumed

US Patent
LigandChemical structure of BindingDB Monomer ID 293492BDBM293492(US10106527, Compound 108 | US9951048, Compound 108...)
Affinity DataEC50:  1nMAssay Description:The GSK3β kinase assay is run using the Ser/Thr 09 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologiesa Div...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293424BDBM293424(US10106527, Compound 142 | US10106527, Compound 14...)
Affinity DataEC50:  1nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293478BDBM293478(US10106527, Compound 92 | US9951048, Compound 92 |...)
Affinity DataEC50:  1nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293637BDBM293637(US10106527, Compound 435 | US9951048, Compound 435...)
Affinity DataEC50:  1nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293593BDBM293593(US10106527, Compound 334 | US9951048, Compound 334...)
Affinity DataEC50:  1nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293582BDBM293582(US10106527, Compound 317 | US9951048, Compound 317...)
Affinity DataEC50:  1.10nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293565BDBM293565(US10106527, Compound 276 | US9951048, Compound 276...)
Affinity DataEC50:  1.10nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293420BDBM293420(US10106527, Compound 6 | US9951048, Compound 6 | U...)
Affinity DataEC50:  1.10nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293452BDBM293452(US10106527, Compound 55 | US9951048, Compound 55 |...)
Affinity DataEC50:  1.10nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293442BDBM293442(US10106527, Compound 28 | US9951048, Compound 28 |...)
Affinity DataEC50:  1.10nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293430BDBM293430(US10106527, Compound 16 | US9951048, Compound 16 |...)
Affinity DataEC50:  1.10nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293620BDBM293620(US10106527, Compound 392 | US9951048, Compound 392...)
Affinity DataEC50:  1.10nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293563BDBM293563(US10106527, Compound 273 | US9951048, Compound 273...)
Affinity DataEC50:  1.10nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293595BDBM293595(US10106527, Compound 336 | US9951048, Compound 336...)
Affinity DataEC50:  1.10nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293643BDBM293643(US10106527, Compound 441 | US9951048, Compound 441...)
Affinity DataEC50:  1.10nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293599BDBM293599(US10106527, Compound 340 | US9951048, Compound 340...)
Affinity DataEC50:  1.20nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293421BDBM293421(US10106527, Compound 7 | US9951048, Compound 7 | U...)
Affinity DataEC50:  1.20nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293612BDBM293612(US10106527, Compound 384 | US9951048, Compound 384...)
Affinity DataEC50:  1.20nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293443BDBM293443(US10106527, Compound 29 | US9951048, Compound 29 |...)
Affinity DataEC50:  1.20nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293424BDBM293424(US10106527, Compound 142 | US10106527, Compound 14...)
Affinity DataEC50:  1.20nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293568BDBM293568(US10106527, Compound 285 | US9951048, Compound 285...)
Affinity DataEC50:  1.20nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293415BDBM293415(US10106527, Compound 145 | US10106527, Compound 1 ...)
Affinity DataEC50:  1.20nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293621BDBM293621(US10106527, Compound 393 | US9951048, Compound 393...)
Affinity DataEC50:  1.20nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293419BDBM293419(US10106527, Compound 5 | US9951048, Compound 5 | U...)
Affinity DataEC50:  1.20nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293545BDBM293545(US10106527, Compound 236 | US9951048, Compound 236...)
Affinity DataEC50:  1.20nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293455BDBM293455(US10106527, Compound 59 | US9951048, Compound 59 |...)
Affinity DataEC50:  1.30nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293425BDBM293425(US10106527, Compound 11 | US9951048, Compound 11 |...)
Affinity DataEC50:  1.30nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293639BDBM293639(US10106527, Compound 437 | US9951048, Compound 437...)
Affinity DataEC50:  1.30nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293636BDBM293636(US10106527, Compound 434 | US9951048, Compound 434...)
Affinity DataEC50:  1.30nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293482BDBM293482(US10106527, Compound 97 | US9951048, Compound 97 |...)
Affinity DataEC50:  1.30nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293416BDBM293416(US10106527, Compound 2 | US9951048, Compound 2 | U...)
Affinity DataEC50:  1.30nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293480BDBM293480(US10106527, Compound 94 | US9951048, Compound 94 |...)
Affinity DataEC50:  1.30nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293560BDBM293560(US10106527, Compound 266 | US9951048, Compound 266...)
Affinity DataEC50:  1.30nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293453BDBM293453(US10106527, Compound 56 | US9951048, Compound 56 |...)
Affinity DataEC50:  1.40nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 293554BDBM293554(US10106527, Compound 253 | US9951048, Compound 253...)
Affinity DataEC50:  1.40nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
US Patent

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