Compile Data Set for Download or QSAR
Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 4246
LigandPNGBDBM33024(SMR000445568 | Punicalin | MLS000697664 | cid_5388...)
Affinity DataIC50: 176nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM51319(MLS000037525 | MLS001401404 | ethyl 2-(7-benzyl-3-...)
Affinity DataIC50: 1.40E+3nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM50056939(NSC-92186 | CHEMBL176570 | Parellic acid, 3 | cid_...)
Affinity DataIC50: 5.45E+3nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM50055659(CHEMBL11252 | 2N-[5-(3-amino-3-iminopropylcarbamoy...)
Affinity DataIC50: 6.37E+3nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM29673(NSC-87509 | CHEMBL172439 | cid_5320418 | 1,4,10-Tr...)
Affinity DataIC50: 8.02E+3nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM50056922(cid_73677 | CHEMBL173530 | 1,4-Dihydroxy-10-methox...)
Affinity DataIC50: 8.74E+3nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM43826(MLS000568202 | 2-[[5-(diethylsulfamoyl)-1-(4-metho...)
Affinity DataIC50: 3.48E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM51310(6,7,12,15,15-pentamethyl-3,10-diazatetracyclo[10.2...)
Affinity DataIC50: 3.71E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56841(cid_3237774 | ethyl 4-{[(2-{[(2Z)-3-methyl-1,3-ben...)
Affinity DataIC50: 4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56845(MLS000051428 | (E)-3-(1-methyl-3-indolyl)-2-(4-met...)
Affinity DataIC50: 4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM43831(5-[(4-fluorophenyl)methyl]-4-oxo-6,7-dihydropyrazo...)
Affinity DataIC50: 4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM43833(SMR000185773 | N''''-(5,5-dimethyl-3-oxocyclohexen...)
Affinity DataIC50: 4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM43835(N-cyclohexyl-5-nitro-2-(1-piperidinyl)benzamide | ...)
Affinity DataIC50: 4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM43836(MLS000580208 | N-(2,5-dimethoxyphenyl)-2-(quinolin...)
Affinity DataIC50: 4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56851(SMR000074755 | cid_1305851 | 2-(1,1-dioxido-3-oxo-...)
Affinity DataIC50: 4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM43838(MLS000438679 | cid_16759689 | 4-O-[5-bromo-2-cyclo...)
Affinity DataIC50: 4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM43837(CMLD004122 | methyl (4S,5R,6R)-1-(2-ethoxy-2-oxoet...)
Affinity DataIC50: 4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56826(4-[morpholin-4-yl(2,2,3,3-tetrafluoropropoxy)phosp...)
Affinity DataIC50: 4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56825(cid_649572 | SMR000006972 | 1-Pyrimidin-2-yl-piper...)
Affinity DataIC50: 4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56864(2-(4-quinazolinylamino)hexanoic acid | SMR00013630...)
Affinity DataIC50: 4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56835(methyl 2-azanyl-5-phenyl-1,3-thiazole-4-carboxylat...)
Affinity DataIC50: 4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56836(MLS000082684 | N-(2-phenyl-1-indolyl)acetamide | N...)
Affinity DataIC50: 4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56839(MLS000054855 | 2-[1,3-bis(oxidanylidene)-3a,4,7,7a...)
Affinity DataIC50: 4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56840(SMR000024795 | MLS000090183 | 2-ethyl-2-methyl-3-o...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56843(S-[2-[[6-fluoranyl-3-(2-methoxyethyl)-1,3-benzothi...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56842(1-{[(5-benzyl-1,3,4-oxadiazol-2-yl)thio]acetyl}ind...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56844(methyl [4-({[2-(1-cyclohexen-1-yl)ethyl]amino}sulf...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56847(5-methyl-N-pyridin-3-yl-thiophene-3-carboxamide | ...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56846(MLS000100276 | 2-[4-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56848(2-(4-methoxyphenyl)-5-(prop-2-enylamino)-1,3-oxazo...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56850(SMR000074911 | N-[5-(1-ethylpropyl)-1,3,4-thiadiaz...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56849(N-{3-[2-(4-methylphenyl)-2-oxoethoxy]phenyl}-2-fur...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56852(N-[4-(1,3-benzoxazol-2-yl)phenyl]-1,3-benzodioxole...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56854(SMR000082144 | cid_2979648 | MLS000066735 | 1-(ben...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56853(cid_877545 | 2-[(1-phenyl-1,2,4-triazol-3-yl)thio]...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56856(1-(4-methoxyphenyl)sulfonyl-3-piperidinecarboxylic...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56855(ethyl 2-(methanesulfonamido)-6-methyl-4,5,6,7-tetr...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56858(1-(2-methylphenyl)-3-(oxolan-2-ylmethyl)urea | cid...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56857(SMR000117995 | MLS000527521 | N'-(2-furanylmethyl)...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56860(2-(2-chlorophenyl)-5-hydroxy-6-nitrochromen-4-one ...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56859(cid_536731 | MLS000547529 | ethyl 2-(acetylamino)-...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56862(cid_1489507 | N-(3-thioxo-3H-1,2,4-dithiazol-5-yl)...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56861(6-(1-pyrrolidinyl)-3-(trifluoromethyl)[1,2,4]triaz...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56863(cid_2967386 | SMR000136212 | 2-[(4-methoxyphenyl)s...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56866(N-[4-(2,6-dimethylpiperidin-1-yl)sulfonylphenyl]-3...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56865(N-{[(4,6-dimethyl-2-pyrimidinyl)amino][(2-propoxyp...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM43823(N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-piperidinos...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM56867(cid_2882343 | SMR000141167 | 1-(1-adamantylcarbony...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM43825(methyl (Z)-3-(3-chloro-2-methylanilino)-2-[3-chlor...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
LigandPNGBDBM43824(N-[(E)-N''''-(1,3-benzothiazol-2-yl)carbamimidoyl]...)
Affinity DataIC50: 8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
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