Compile Data Set for Download or QSAR
Report error Found 47 Enz. Inhib. hit(s) with all data for entry = 3484
LigandChemical structure of BindingDB Monomer ID 33114BDBM33114([2-(6-amino-1-benzyl-3-methyl-2,4-dioxopyrimidin-5...)
Affinity DataIC50: 1.34E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35479BDBM35479(cid_9547735 | [2-(4-amino-1-benzyl-3-methyl-2,6-di...)
Affinity DataIC50: 1.69E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35463BDBM35463(CC-PMLSC-DMA-P138 | [2-[4-azanyl-1,3-dimethyl-2,6-...)
Affinity DataIC50: 2.06E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35484BDBM35484([2-[6-amino-1-(cyclopropylmethyl)-3-methyl-2,4-dio...)
Affinity DataIC50: 2.46E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35480BDBM35480(cid_9547736 | 2-cyclopropyl-4-quinolinecarboxylic ...)
Affinity DataIC50: 2.89E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35477BDBM35477([2-(4-amino-1-benzyl-3-methyl-2,6-dioxopyrimidin-5...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35478BDBM35478([2-[6-azanyl-1-methyl-2,4-bis(oxidanylidene)-3-(ph...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35481BDBM35481(cid_9547737 | [2-(4-amino-1-benzyl-3-methyl-2,6-di...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35482BDBM35482(cid_9547738 | [2-[4-azanyl-1-methyl-3-(2-methylpro...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35483BDBM35483(cid_9547739 | CC-PMLSC-DMA-P164 | 6-amino-5-(2-chl...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35485BDBM35485([2-[6-amino-1-(cyclopropylmethyl)-3-methyl-2,4-dio...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35441BDBM35441(6-amino-5-(2-chloro-1-oxoethyl)-1,3-dimethylpyrimi...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35442BDBM35442([2-[4-azanyl-1,3-dimethyl-2,6-bis(oxidanylidene)py...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35443BDBM35443(6-amino-5-(2-chloro-1-oxoethyl)-3-methyl-1-(2-meth...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35444BDBM35444(2-phenyl-4-quinolinecarboxylic acid [2-(4-amino-1,...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35445BDBM35445(2-phenyl-4-quinolinecarboxylic acid [2-[4-amino-1-...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35446BDBM35446(2,8-bis(trifluoromethyl)-1H-quinolin-4-one | CC-PM...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35447BDBM35447(cid_10853 | (phenylmethyl)urea | 1-(phenylmethyl)u...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35448BDBM35448(CC-PMLSC-DMA-P108 | 4-bromanyl-2,8-bis(trifluorome...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35449BDBM35449(6-amino-1-benzylpyrimidine-2,4-dione | 6-amino-1-(...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35450BDBM35450(N'-[2,6-dioxo-3-(phenylmethyl)-4-pyrimidinyl]-N,N-...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35451BDBM35451(cid_9547712 | 2-(trifluoromethyl)quinoline-4-carbo...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35452BDBM35452(2,8-bis(trifluoromethyl)-4-quinolinecarboxylic aci...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35453BDBM35453(CHEMBL150924 | 2-(2-furanyl)-4-quinolinecarboxylic...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35454BDBM35454(2-cyclopropyl-4-quinolinecarboxylic acid | cid_275...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35379BDBM35379([2-[4-azanyl-1-methyl-3-(2-methylpropyl)-2,6-bis(o...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35455BDBM35455(1-(cyclopropylmethyl)urea | cid_9547713 | CC-PMLSC...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35456BDBM35456(N,N-dimethyl-N'-(3-methyl-2,6-dioxo-4-pyrimidinyl)...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35457BDBM35457(N,N-dimethyl-N'-[1-methyl-2,6-bis(oxidanylidene)-3...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35458BDBM35458(CC-PMLSC-DMA-P130 | cid_9547716 | 2-cyano-N-(cyclo...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35459BDBM35459(cid_9547717 | N,N-dimethyl-N'-[3-methyl-2,6-bis(ox...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35460BDBM35460(cid_9547718 | 6-amino-1-(cyclopropylmethyl)pyrimid...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35461BDBM35461(cid_1649246 | 6-amino-3-methyl-1-(phenylmethyl)pyr...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35462BDBM35462(6-amino-3-benzyl-1-methylpyrimidine-2,4-dione | ci...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35464BDBM35464(CC-PMLSC- DMA-P139 | cid_9547720 | N'-[3-(cyclopro...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35465BDBM35465([2-(4-amino-1,3-dimethyl-2,6-dioxopyrimidin-5-yl)-...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35466BDBM35466([2-[4-azanyl-1-methyl-3-(2-methylpropyl)-2,6-bis(o...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35467BDBM35467(N'-[3-(cyclopropylmethyl)-1-methyl-2,6-bis(oxidany...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35468BDBM35468(CC-PMLSC-DMA-P143 | 6-azanyl-5-(2-chloranylethanoy...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35469BDBM35469(2-(trifluoromethyl)-4-quinolinecarboxylic acid [2-...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35470BDBM35470(CC-PMLSC-DMA-P146 | cid_9547725 | [2-[4-azanyl-1,3...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35471BDBM35471(2-phenyl-4-quinolinecarboxylic acid [2-[4-amino-1-...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35472BDBM35472(6-azanyl-5-(2-chloranylethanoyl)-1-methyl-3-(pheny...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35473BDBM35473(cid_9547728 | CC-PMLSC-DMA-P152 | 2,8-bis(trifluor...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35474BDBM35474(cid_9547729 | CC-PMLSC-DMA-P154 | [2-[4-azanyl-1-m...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35475BDBM35475(CC-PMLSC-DMA-P155 | [2-(6-amino-1-benzyl-3-methyl-...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay
LigandChemical structure of BindingDB Monomer ID 35476BDBM35476(CC-PMLSC-DMA-P157 | [2-(6-amino-1-benzyl-3-methyl-...)
Affinity DataIC50: 5.00E+4nMpH: 7.0 T: 2°CAssay Description:The MKP-1 dose response assay SAR support Assay - has been developed to test the activity of a series Analog compounds synthesized by the PMLSC Chemi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details
PCBioAssay