Reaction Details
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Cell Reactant:
Cyclin-dependent protein kinase 2 variant (CDK2 C118L/A144C)
Syringe Reactant:
BDBM154576
Meas. Tech.:
Enzyme Inhibition
Entry Date.:
10/15/15
ΔG°:
-10.62±0 (kcal/mole)
pH:
7.5±0
Temperature:
288.15±0 (K)
ΔH° :
-18.21±n/a (kJ/mole)
ΔHobs :
-18.04±0 (kJ/mole)
ΔS° :
-0.03±0 (kJ/mole-K)
Citation
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More Info.:
Cell React
Name:
Cyclin-dependent kinase 2 [C118L,A144C]
Synonyms:
CDK2 | CDK2_HUMAN | CDKN2 | Cyclin-dependent protein kinase 2 variant (CDK2 C118L/A144C)
Type:
Protein
Mol. Mass.:
33980.25
Organism:
Homo sapiens (Human)
Description:
CDK2 mutant (C118L/A144C)
Residue:
298
Sequence:
MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFLHSHRVLHRDLKPQNLLINTEGAIKLCDFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL