Reaction Details
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Target
Isocitrate dehydrogenase [NADP] cytoplasmic [R132G]
Ligand
BDBM50506474
Substrate
n/a
Meas. Tech.
Biochemical Assay
IC50
<50.0±n/a nM
Citation
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More Info.:
Target
Name:
Isocitrate dehydrogenase [NADP] cytoplasmic [R132G]
Synonyms:
IDH1 | IDHC_HUMAN | Isocitrate dehydrogenase 1 mutant (R132G) | PICD
Type:
Protein
Mol. Mass.:
46561.14
Organism:
Homo sapiens (Human)
Description:
R132G mutant
Residue:
414
Sequence:
MSKKISGGSVVEMQGDEMTRIIWELIKEKLIFPYVELDLHSYDLGIENRDATNDQVTKDAAEAIKKHNVGVKCATITPDEKRVEEFKLKQMWKSPNGTIRNILGGTVFREAIICKNIPRLVSGWVKPIIIGGHAYGDQYRATDFVVPGPGKVEITYTPSDGTQKVTYLVHNFEEGGGVAMGMYNQDKSIEDFAHSSFQMALSKGWPLYLSTKNTILKKYDGRFKDIFQEIYDKQYKSQFEAQKIWYEHRLIDDMVAQAMKSEGGFIWACKNYDGDVQSDSVAQGYGSLGMMTSVLVCPDGKTVEAEAAHGTVTRHYRMYQKGQETSTNPIASIFAWTRGLAHRAKLDNNKELAFFANALEEVSIETIEAGFMTKDLAACIKGLPNVQRSDYLNTFEFMDKLGENLKIKLAQAKL