Reaction Details Report a problem with these data
Target
Chitinase-3-like protein 1
Ligand
BDBM616592
Substrate
n/a
Meas. Tech.
YKL-40: HS Assay
IC50
<100±n/a nM
Citation
Krzeminski, L; Czestkowski, W; Mazur, M; Andryianau, G; Olejniczak, S; Piotrowicz, MC; Koralewski, R; Pluta, E; Matyszewski, K; Kowalski, M; Dymek, B; Koziel, R; Olczak, J; Golebiowski, A; Bartoszewicz, A; Krysztofiak, K YKL-40 INHIBITORS AND THEIR THERAPEUTIC APPLICATIONS US Patent US20230278996 Publication Date 9/7/2023
More Info.:
Target
Name:
Chitinase-3-like protein 1
Synonyms:
39 kDa synovial protein | CGP-39 | Cartilage glycoprotein 39 | GP-39 | YKL-40 | hCGP-39
Type:
Protein
Mol. Mass.:
42634.54
Organism:
Human
Description:
P36222
Residue:
383
Sequence:
MGVKASQTGFVVLVLLQCCSAYKLVCYYTSWSQYREGDGSCFPDALDRFLCTHIIYSFANISNDHIDTWEWNDVTLYGMLNTLKNRNPNLKTLLSVGGWNFGSQRFSKIASNTQSRRTFIKSVPPFLRTHGFDGLDLAWLYPGRRDKQHFTTLIKEMKAEFIKEAQPGKKQLLLSAALSAGKVTIDSSYDIAKISQHLDFISIMTYDFHGAWRGTTGHHSPLFRGQEDASPDRFSNTDYAVGYMLRLGAPASKLVMGIPTFGRSFTLASSETGVGAPISGPGIPGRFTKEAGTLAYYEICDFLRGATVHRILGQQVPYATKGNQWVGYDDQESVKSKVQYLKDRQLAGAMVWALDLDDFQGSFCGQDLRFPLTNAIKDALAAT