Reaction Details
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Target
Gamma-aminobutyric acid receptor subunit beta-1
Ligand
BDBM625660
Substrate
n/a
Meas. Tech.
Steroid Inhibition of TBPS Binding
IC50
<100±n/a nM
Citation
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More Info.:
Target
Name:
Gamma-aminobutyric acid receptor subunit beta-1
Synonyms:
GABA(A) receptor subunit beta-1
Type:
Protein
Mol. Mass.:
54082.33
Organism:
Rat
Description:
P15431
Residue:
474
Sequence:
MWTVQNRESLGLLSFPVMVAMVCCAHSSNEPSNMSYVKETVDRLLKGYDIRLRPDFGGPPVDVGMRIDVASIDMVSEVNMDYTLTMYFQQSWKDKRLSYSGIPLNLTLDNRVADQLWVPDTYFLNDKKSFVHGVTVKNRMIRLHPDGTVLYGLRITTTAACMMDLRRYPLDEQNCTLEIESYGYTTDDIEFYWNGGEGAVTGVNKIELPQFSIVDYKMVSKKVEFTTGAYPRLSLSFRLKRNIGYFILQTYMPSTLITILSWVSFWINYDASAARVALGITTVLTMTTISTHLRETLPKIPYVKAIDIYLMGCFVFVFLALLEYAFVNYIFFGKGPQKKGASKQDQSANEKNKLEMNKVQVDAHGNILLSTLEIRNETSGSEVLTGVSDPKATMYSYDSASIQYRKPLSSREGFGRGLDRHGVPGKGRIRRRASQLKVKIPDLTDVNSIDKWSRMFFPITFSLFNVVYWLYYVH