Reaction Details Report a problem with these data
Target
Bisphosphoglycerate mutase
Ligand
BDBM632770
Substrate
n/a
Meas. Tech.
BPGM Synthase Assay
IC50
99.0±n/a nM
Citation
Desai, K; Fang, Z; Guertin, K; Hong, V; Jiang, JZ; Lim, S; Munson, M CARBOXYLIC ACID-CONTAINING COMPOUNDS AS MODULATORS OF BIS-PHOSPHOGLYCERATE MUTASE FOR THE TREATMENT OF SICKLE CELL DISEASE US Patent US20230348450 Publication Date 11/2/2023
More Info.:
Target
Name:
Bisphosphoglycerate mutase
Synonyms:
2,3-bisphosphoglycerate mutase, erythrocyte | 2,3-bisphosphoglycerate synthase | 2,3-diphosphoglycerate mutase | 5.4.2.11 | 5.4.2.4 | BPG-dependent PGAM | BPGM | PMGE_HUMAN
Type:
PROTEIN
Mol. Mass.:
30004.85
Organism:
Homo sapiens
Description:
ChEMBL_120651
Residue:
259
Sequence:
MSKYKLIMLRHGEGAWNKENRFCSWVDQKLNSEGMEEARNCGKQLKALNFEFDLVFTSVLNRSIHTAWLILEELGQEWVPVESSWRLNERHYGALIGLNREQMALNHGEEQVRLWRRSYNVTPPPIEESHPYYQEIYNDRRYKVCDVPLDQLPRSESLKDVLERLLPYWNERIAPEVLRGKTILISAHGNSSRALLKHLEGISDEDIINITLPTGVPILLELDENLRAVGPHQFLGDQEAIQAAIKKVEDQGKVKQAKK