Reaction Details Report a problem with these data
Target
Sigma intracellular receptor 2
Ligand
BDBM312185
Substrate
n/a
Meas. Tech.
Receptor Assay
Ki
0.560±0.12 nM
Citation
McCurdy, CR; Mesangeau, C; Chin, FT; James, ML; Shen, B; Gambhir, S Highly selective sigma receptor radioligands US Patent US9604926 Publication Date 3/28/2017
More Info.:
Target
Name:
Sigma intracellular receptor 2
Synonyms:
S2r | SGMR2_MOUSE | Sigma-2 receptor | Sigma2 receptor | Tmem97 | Transmembrane protein 97
Type:
n/a
Mol. Mass.:
20818.69
Organism:
Mouse
Description:
Q8VD00
Residue:
176
Sequence:
MGALAARRCVEWLLGLYFVSHIPITLFIDLQAVLPPELYPQEFSNLLRWYSKEFKDPLMQEPPVWFKSFLLCELVFQLPFFPIAAYAFFKGSCRWIRIPAIIYAAHTITTLIPILYTLLFEDFSKAVAFKGQRPESFRERLTLVGVYAPYLIIPLILLLFMLRNPYYKYEEKRKKK