Reaction Details Report a problem with these data
Target
Ubiquitin carboxyl-terminal hydrolase isozyme L5
Ligand
BDBM50069762
Substrate
n/a
Meas. Tech.
Fluorometric Ub-AMC Hydrolysis Assay
pH
7.5±n/a
Temperature
298.15±n/a K
IC50
>114000±n/a nM
Comments
extracted
Citation
Ott, CA; Baljinnyam, B; Zakharov, AV; Jadhav, A; Simeonov, A; Zhuang, Z Cell Lysate-Based AlphaLISA Deubiquitinase Assay Platform for Identification of Small Molecule Inhibitors. ACS Chem Biol 12:2399-2407 (2017) [PubMed] Article
More Info.:
Target
Name:
Ubiquitin carboxyl-terminal hydrolase isozyme L5
Synonyms:
CGI-70 | UCH-L5 | UCH37 | UCHL5 | UCHL5_HUMAN | Ubiquitin C-terminal hydrolase UCH37 | Ubiquitin carboxyl-terminal hydrolase isozyme L5 | Ubiquitin thioesterase L5
Type:
PROTEIN
Mol. Mass.:
37597.89
Organism:
Homo sapiens (Human)
Description:
ChEMBL_109575
Residue:
329
Sequence:
MTGNAGEWCLMESDPGVFTELIKGFGCRGAQVEEIWSLEPENFEKLKPVHGLIFLFKWQPGEEPAGSVVQDSRLDTIFFAKQVINNACATQAIVSVLLNCTHQDVHLGETLSEFKEFSQSFDAAMKGLALSNSDVIRQVHNSFARQQMFEFDTKTSAKEEDAFHFVSYVPVNGRLYELDGLREGPIDLGACNQDDWISAVRPVIEKRIQKYSEGEIRFNLMAIVSDRKMIYEQKIAELQRQLAEEEPMDTDQGNSMLSAIQSEVAKNQMLIEEEVQKLKRYKIENIRRKHNYLPFIMELLKTLAEHQQLIPLVEKAKEKQNAKKAQETK