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Target
15-hydroxyprostaglandin dehydrogenase [NAD(+)]
Ligand
BDBM347359
Substrate
n/a
Meas. Tech.
In Vitro Assay
IC50
0.760±n/a nM
Citation
Markowitz, S; Willson, JK; Posner, BA; Ready, J; Zhang, Y; Tai, H; Antczak, M; Gerson, S; Bae, K; Yang, SY; Desai, A Compositions and methods of modulating 15-PGDH activity US Patent US9790233 Publication Date 10/17/2017
More Info.:
Target
Name:
15-hydroxyprostaglandin dehydrogenase [NAD(+)]
Synonyms:
15-PGDH | 15-hydroxyprostaglandin dehydrogenase [NAD+] | HPGD | PGDH1 | PGDH_HUMAN | Prostaglandin dehydrogenase 1 (15-PGDH) | SDR36C1
Type:
Enzyme
Mol. Mass.:
28974.46
Organism:
Human
Description:
P15428
Residue:
266
Sequence:
MHVNGKVALVTGAAQGIGRAFAEALLLKGAKVALVDWNLEAGVQCKAALDEQFEPQKTLFIQCDVADQQQLRDTFRKVVDHFGRLDILVNNAGVNNEKNWEKTLQINLVSVISGTYLGLDYMSKQNGGEGGIIINMSSLAGLMPVAQQPVYCASKHGIVGFTRSAALAANLMNSGVRLNAICPGFVNTAILESIEKEENMGQYIEYKDHIKDMIKYYGILDPPLIANGLITLIEDDALNGAIMKITTSKGIHFQDYDTTPFQAKTQ